SCHEMBL7439062

SCHEMBL7439062

CCCN(CCC)C1Cc2cc3cc[nH]c3cc2C1

nearest known ligand 0.82

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FYN P06241 2/20 0.54
DRD3 P35462 1/20 0.53
HTR1D P28221 4/20 0.52
HTR1B P28222 3/20 0.52
ALDH1A1 P00352 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
ALOX15 P16050 1/20 0.51
MAPK1 P28482 1/20 0.51
HTR1A P08908 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7435180 0.91 HTR1D (0.62) FYNDRD3HTR1DHTR1BCYP2D6
SCHEMBL7441326 0.90 HTR1D (0.58) FYNDRD3HTR1DHTR1BALDH1A1
SCHEMBL7443837 0.87 HTR1D (0.59) FYNDRD3HTR1DHTR1B
SCHEMBL7443957 0.87 HTR1D (0.48) FYNDRD3HTR1DHTR1B
SCHEMBL7442744 0.75 HTR1D (0.81) HTR1DHTR1B
SCHEMBL7441299 0.74 HTR1D (0.53) FYNDRD3HTR1DHTR1BHTR1A
SCHEMBL7439287 0.73 HTR1D (0.49) DRD3HTR1DHTR1BHTR1A
SCHEMBL7447452 0.72 DRD2 (0.55) DRD3HTR1DHTR1BHTR1A
SCHEMBL7447457 0.72 DRD2 (0.55) DRD3HTR1DHTR1BHTR1A
SCHEMBL8693035 0.72 FYN (0.70) FYNDRD3ALDH1A1CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0690843-B1 Formyl- or cyano- substituted indole derivatives having dopaminergic activity UPJOHN CO (US) 2000-08-30 EP disclosed
US-5639778-A TREATING CENTRAL NERVOUS SYSTEM DISORDERS PHARMACIA & UPJOHN COMPANY (US) 1997-06-17 US disclosed
EP-0690843-A1 INDOLETETRALINS HAVING DOPAMINERGIC ACTIVITY PHARMACIA & UPJOHN COMPANY (US) 1996-01-10 EP disclosed
WO-1994021608-A1 INDOLETETRALINS HAVING DOPAMINERGIC ACTIVITY THE UPJOHN COMPANY (US) 1994-09-29 WO disclosed