SCHEMBL7439162

SCHEMBL7439162

O=C(Nc1ccccc1)c1ccccc1S(=O)(=O)O

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 2/20 0.73
ALDH1A1 P00352 2/20 0.59
MEN1 O00255 6/20 0.58
KMT2A Q03164 6/20 0.58
HPGD P15428 3/20 0.58
KDM4E B2RXH2 1/20 0.58
LMNA P02545 1/20 0.58
TP53 P04637 1/20 0.58
HTT P42858 1/20 0.58
HSD17B10 Q99714 1/20 0.58
TDP1 Q9NUW8 3/20 0.56
CYP3A4 P08684 2/20 0.54
CYP2C9 P11712 2/20 0.54
METAP2 P50579 1/20 0.54
ALOX12 P18054 1/20 0.54
CHRNB2 P17787 1/20 0.54
CHRNB4 P30926 1/20 0.54
CHRNA3 P32297 1/20 0.54
CHRNA4 P43681 1/20 0.54
POLB P06746 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27430115 0.84 CA1 (0.68) BCAT2ALDH1A1MEN1KMT2ALMNA
SCHEMBL6552449 0.84 BCAT2 (0.71) BCAT2ALDH1A1MEN1KMT2AHPGD
SCHEMBL8379611 0.84 BCAT2 (0.71) BCAT2ALDH1A1MEN1KMT2AHPGD
SCHEMBL16102705 0.84 BCAT2 (1.00) BCAT2ALDH1A1MEN1KMT2AHPGD
SCHEMBL12700257 0.83 BCAT2 (0.52) BCAT2ALDH1A1MEN1KMT2ALMNA
SCHEMBL5187712 0.83 BCAT2 (0.69) BCAT2ALDH1A1MEN1KMT2AHPGD
SCHEMBL7224833 0.81 BCAT2 (0.77) BCAT2ALDH1A1MEN1KMT2AHPGD
SCHEMBL437231 0.80 ALDH1A1 (0.87) BCAT2ALDH1A1MEN1KMT2AHPGD
SCHEMBL7130887 0.79 BCAT2 (0.63) BCAT2ALDH1A1MEN1KMT2AHPGD
SCHEMBL11266257 0.78 ALDH1A1 (0.83) BCAT2ALDH1A1MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed