SCHEMBL437231

SCHEMBL437231

O=C(Nc1ccccc1)c1ccccc1C(=O)Nc1ccccc1

nearest known ligand 0.87

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.87
MEN1 O00255 7/20 0.76
KMT2A Q03164 7/20 0.76
HPGD P15428 2/20 0.76
TP53 P04637 2/20 0.76
KDM4E B2RXH2 1/20 0.76
LMNA P02545 1/20 0.76
HTT P42858 1/20 0.76
HSD17B10 Q99714 1/20 0.76
TDP1 Q9NUW8 3/20 0.73
METAP2 P50579 1/20 0.70
CYP3A4 P08684 1/20 0.70
CYP2C9 P11712 1/20 0.70
ALOX12 P18054 1/20 0.70
CHRNB2 P17787 1/20 0.70
CHRNB4 P30926 1/20 0.70
CHRNA3 P32297 1/20 0.70
CHRNA4 P43681 1/20 0.70
BCAT2 O15382 2/20 0.66
POLB P06746 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11266259 0.98 ALDH1A1 (0.83) ALDH1A1MEN1KMT2AHPGDTP53
SCHEMBL11266257 0.98 ALDH1A1 (0.83) ALDH1A1MEN1KMT2AHPGDTP53
SCHEMBL1991348 0.93 ALDH1A1 (1.00) ALDH1A1MEN1KMT2AHPGDTP53
SCHEMBL45299 0.93 ALDH1A1 (1.00) ALDH1A1MEN1KMT2AHPGDTP53
SCHEMBL1991352 0.89 ALDH1A1 (0.71) ALDH1A1MEN1KMT2AHPGDTP53
SCHEMBL9853958 0.89 ALDH1A1 (0.71) ALDH1A1MEN1KMT2AHPGDTP53
SCHEMBL29024967 0.89 ALDH1A1 (0.71) ALDH1A1MEN1KMT2AHPGDTP53
SCHEMBL18784684 0.89 ALDH1A1 (0.71) ALDH1A1MEN1KMT2AHPGDTP53
SCHEMBL16634926 0.89 ALDH1A1 (0.71) ALDH1A1MEN1KMT2AHPGDTP53
SCHEMBL1533636 0.89 ALDH1A1 (0.71) ALDH1A1MEN1KMT2AHPGDTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 307 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114481448-A Nanofiber membrane and preparation method and application thereof 中国石油化工股份有限公司 2022-05-13 CN claimed
US-20150265610-A1 COMBINATIONS FOR THE TREATMENT OF DISEASES INVOLVING CELL PROLIFERATION, MIGRATION OR APOPTOSIS OF MYELOMA CELLS, OR ANGIOGENESIS BOEHRINGER INGELHEIM INT (DE) 2015-09-24 US claimed
EP-2826480-A1 Combinations for the treatment of diseases involving cell proliferation, migration or apoptosis of myeloma cells, or angiogenesis Boehringer Ingelheim International GmbH (DE) 2015-01-21 EP claimed
EP-2124951-B1 5-CYAN0-4- (PYRROLO[2, 3B]PYRIDINE-3-YL) -PYRIMIDINE DERIVATIVES USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMA (US) 2014-05-21 EP claimed
US-20140057898-A1 COMBINATIONS FOR THE TREATMENT OF DISEASES INVOLVING CELL PROLIFERATION, MIGRATION OR APOPTOSIS OF MYELOMA CELLS, OR ANGIOGENESIS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-02-27 US claimed
US-8247421-B2 5-cyano-4-(pyrrolo [2,3B] pyridine-3-yl)-pyrimidine derivatives useful as protein kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-08-21 US claimed
EP-2409705-A1 Combinations for the treatment of diseases involving cell proliferation, migration or apoptosis of myeloma cells or angiogenesis BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-25 EP claimed
EP-2361626-A1 Combinations for the treatment of diseases involving cell proliferation, migration or apoptosis of myeloma cells, or angiogenesis BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-08-31 EP claimed
EP-2359829-A1 Combinations for the treatment of diseases involving cell proliferation, migration or apoptosis of myeloma cells, or angiogenesis BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-08-24 EP claimed
US-20110171289-A1 COMBINATIONS FOR THE TREATMENT OF DISEASES INVOLVING CELL PROLIFERATION, MIGRATION OR APOPTOSIS OF MYELOMA CELLS, OR ANGIOGENESIS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-14 US claimed
US-7223851-B2 Nucleic acid-binding polymers GENERAL DYNAMICS ADVANCED INFORMATION SYSTEMS, INC. (US) 2007-05-29 US claimed
JP-2006524634-A 2006-11-02 JP claimed
CN-1780627-A Combinations for the treatment of diseases involving cell proliferation, migration or apoptosis of myeloma cells or vascular proliferation BOEHRINGER INGELHEIM INT (DE) 2006-05-31 CN claimed
US-20060058311-A1 Combinations for the treatment of diseases involving cell proliferation BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-03-16 US claimed
WO-2006018182-A1 COMBINATIONS FOR THE TREATMENT OF DISEASES INVOLVING CELL PROLIFERATION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-02-23 WO claimed
EP-1622619-A2 COMBINATIONS FOR THE TREATMENT OF DISEASES INVOLVING CELL PROLIFERATION, MIGRATION OR APOPTOSIS OF MYELOMA CELLS, OR ANGIOGENESIS Boehringer Ingelheim International GmbH (DE) 2006-02-08 EP claimed
US-20050043233-A1 Combinations for the treatment of diseases involving cell proliferation, migration or apoptosis of myeloma cells or angiogenesis BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-02-24 US claimed
WO-2004096224-A2 COMBINATIONS FOR THE TREATMENT OF DISEASES INVOLVING CELL PROLIFERATION, MIGRATION OR APOPTOSIS OF MYELOMA CELLS, OR ANGIOGENESIS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2004-11-11 WO claimed
US-20040157217-A1 Nucleic acid-binding polymers VERIDIAN SYSTEMS DIVISION 2004-08-12 US claimed
US-4405678-A Protected vapor-deposited metal layers MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1983-09-20 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140057898-A1 COMBINATIONS FOR THE TREATMENT OF DISEASES INVOLVING CELL PROLIFERATION, MIGRATION OR APOPTOSIS OF MYELOMA CELLS, OR ANGIOGENESIS BAX, BCL2, VEGFA ALDH1A1 2021/4885MEN1 820/4885KMT2A 4330/4885
US-20110171289-A1 COMBINATIONS FOR THE TREATMENT OF DISEASES INVOLVING CELL PROLIFERATION, MIGRATION OR APOPTOSIS OF MYELOMA CELLS, OR ANGIOGENESIS BAX, BCL2, VEGFA ALDH1A1 2021/4885MEN1 820/4885KMT2A 4330/4885
US-20060058311-A1 Combinations for the treatment of diseases involving cell proliferation CCNA1, MKI67, CCNA2 ALDH1A1 1053/4885MEN1 231/4885KMT2A 3566/4885
US-20150265610-A1 COMBINATIONS FOR THE TREATMENT OF DISEASES INVOLVING CELL PROLIFERATION, MIGRATION OR APOPTOSIS OF MYELOMA CELLS, OR ANGIOGENESIS BAX, BCL2, VEGFA ALDH1A1 2021/4885MEN1 820/4885KMT2A 4330/4885
US-20050043233-A1 Combinations for the treatment of diseases involving cell proliferation, migration or apoptosis of myeloma cells or angiogenesis BAX, BCL2, CXCL12 ALDH1A1 2154/4885MEN1 759/4885KMT2A 4366/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.