SCHEMBL7439170

SCHEMBL7439170

CC(C)CC(C(=O)NS(=O)(=O)CC#N)c1csc(N(C)C)n1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSK P43235 11/20 0.47
UCHL1 P09936 1/20 0.33
CTSL P07711 7/20 0.32
CTSS P25774 8/20 0.32
CTSB P07858 4/20 0.32
PDE5A O76074 1/20 0.32
PDE1A P54750 1/20 0.32
PDE1B Q01064 1/20 0.32
PDE1C Q14123 1/20 0.32
FFAR2 O15552 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718663 0.83 CTSK (0.65) CTSKCTSLCTSSCTSB
SCHEMBL7434589 0.65 CTSK (0.57) CTSKCTSLCTSSCTSB
SCHEMBL4714573 0.64 CTSK (1.00) CTSKCTSLCTSSCTSB
SCHEMBL4715211 0.63 CTSK (0.85) CTSKCTSLCTSSCTSB
SCHEMBL13379959 0.61 UCHL1 (0.41) UCHL1MEN1KMT2A
SCHEMBL7439178 0.60 ALDH1A1 (0.32) UCHL1MEN1KMT2A
SCHEMBL13746373 0.59 MEN1 (0.40) UCHL1MEN1KMT2A
SCHEMBL4714808 0.55 CTSK (0.66) CTSKCTSLCTSSCTSB
SCHEMBL11991384 0.54 MEN1 (0.47) MEN1KMT2A
SCHEMBL21229023 0.53 MEN1 (0.57) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001049288-A9 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2001-10-25 WO disclosed