SCHEMBL7439352

SCHEMBL7439352

O=C1CCCc2c1ccc(=O)n2CCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CSNK2A2 P19784 5/20 0.56
CSNK2B P67870 5/20 0.56
CSNK2A1 P68400 5/20 0.56
ABCG2 Q9UNQ0 5/20 0.56
BRD4 O60885 1/20 0.50
HPGD P15428 1/20 0.48
SIGMAR1 Q99720 1/20 0.45
ALB P02768 1/20 0.44
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
MAOA P21397 3/20 0.44
MAOB P27338 3/20 0.44
SLC6A3 Q01959 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7448030 0.85 BRD4 (0.63) CSNK2A2CSNK2BCSNK2A1ABCG2BRD4
SCHEMBL7445206 0.79 BRD4 (0.45) CSNK2A1BRD4HPGDLMNA
SCHEMBL9802743 0.79 HPGD (0.46) CSNK2A2CSNK2BCSNK2A1ABCG2BRD4
SCHEMBL9803168 0.77 BRD4 (0.43) CSNK2A2CSNK2BCSNK2A1ABCG2BRD4
SCHEMBL9803012 0.75 HPGD (0.40) CSNK2A2CSNK2BCSNK2A1ABCG2BRD4
SCHEMBL9802730 0.75 BRD4 (0.47) CSNK2A1BRD4HPGDMAOAMAOB
SCHEMBL9802740 0.75 HPGD (0.51) BRD4HPGDMAOAMAOBLMNA
SCHEMBL7430749 0.74 NPC1 (0.44) CSNK2A1BRD4HPGDLMNA
SCHEMBL9803346 0.73 ALDH1A1 (0.42) CSNK2A2CSNK2BCSNK2A1ABCG2BRD4
SCHEMBL261530 0.72 CSNK2B (1.00) CSNK2A2CSNK2BCSNK2A1ABCG2ALB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6472408-B1 TWO 5- AMINO-5,6,7,8-TETRAHYDROQUINOLINE FRAGMENTS JOINED TOGETHER BY A DIVALENT LINKING GROUP; CHOLINESTERASE INHIBITORS THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (HK) 2002-10-29 US disclosed
US-20020156096-A1 Dimeric compounds HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY, THE (HK) 2002-10-24 US disclosed
EP-0489379-B1 5-amino-5,6,7,8-tetrahydroquinolines and related compounds, a process for their preparation and their use as medicaments HOECHST MARION ROUSSEL INC (US) 1998-07-15 EP disclosed
US-5310914-A Imination, reduction HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-05-10 US disclosed
US-5216164-A Used for relieving memory dysfunction such as Alzheimer's disease HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-06-01 US disclosed
EP-0489379-A1 5-amino-5,6,7,8-tetrahydroquinolines and related compounds, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-06-10 EP disclosed
US-5110815-A Alzheimer's disease HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-05-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020156096-A1 Dimeric compounds ACHE, BCHE, CHRNA5 CSNK2A2 1619/4885CSNK2B 1974/4885CSNK2A1 2297/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.