SCHEMBL7440283

SCHEMBL7440283

CCCCNC(=O)Nc1c(OC(=O)N(CC)CC)nc(C)c2cc(OC)c(OC)cc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.44
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
LCK P06239 2/20 0.39
HSD17B10 Q99714 3/20 0.37
GAA P10253 2/20 0.37
APAF1 O14727 1/20 0.37
TDP2 O95551 1/20 0.37
MAPK1 P28482 1/20 0.37
CASP3 P42574 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
PKM P14618 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
PDE10A Q9Y233 1/20 0.37
QPCT Q16769 3/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447594 0.95 LCK (0.41) KDRALDH1A1KDM4ELCKHSD17B10
SCHEMBL7436056 0.89 KDR (0.42) KDRALDH1A1KDM4ELCKHSD17B10
SCHEMBL7446891 0.83 LMNA (0.41) ALDH1A1KDM4EHSD17B10LMNAMAPT
SCHEMBL7435587 0.82 QPCT (0.38) KDRALDH1A1HSD17B10GAAAPAF1
SCHEMBL9831559 0.81 KDR (0.49) KDRALDH1A1KDM4ELCKHSD17B10
Water SCHEMBL10786986 0.80 KDR (0.48) KDRALDH1A1KDM4ELCKHSD17B10
Water SCHEMBL10786992 0.80 KDR (0.48) KDRALDH1A1KDM4ELCKHSD17B10
SCHEMBL7426725 0.76 LMNA (0.43) ALDH1A1KDM4EGAALMNAMAPT
SCHEMBL7440286 0.73 LMNA (0.35) ALDH1A1KDM4EHSD17B10GAALMNA
SCHEMBL7441183 0.72 LMNA (0.39) ALDH1A1KDM4ECASP3SENP8SENP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4880817-A O-functionalized derivatives of substituted isoquinolin-3-ols having cardiotonic and/or phosphodiesterase fraction III inhibiting properties and/or renal vasodilating properties ORTHO PHARMACEUTICAL CORPORATION (US) 1989-11-14 US claimed
US-4880817-A O-functionalized derivatives of substituted isoquinolin-3-ols having cardiotonic and/or phosphodiesterase fraction III inhibiting properties and/or renal vasodilating properties ORTHO PHARMACEUTICAL CORPORATION (US) 1989-11-14 US disclosed