SCHEMBL7440286

SCHEMBL7440286

CCCCN(C(N)=O)c1c(OC(=O)N(CC)CC)nc(C)c2cc(OC)c(OC)cc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
TSPO P30536 5/20 0.33
ALOX15 P16050 1/20 0.33
KDM4E B2RXH2 4/20 0.32
ALDH1A1 P00352 2/20 0.32
NPC1 O15118 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 3/20 0.32
QPCT Q16769 1/20 0.32
CRHR1 P34998 1/20 0.31
MEN1 O00255 2/20 0.31
MAPT P10636 1/20 0.31
CASP1 P29466 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447598 0.94 TSPO (0.34) LMNATSPOKDM4ENPC1RAB9A
SCHEMBL7436061 0.88 KMT2A (0.32) LMNAKDM4ENPC1GLAKMT2A
SCHEMBL9831575 0.82 KDM4E (0.36) LMNACYP3A4CYP2D6KDM4EALDH1A1
Water SCHEMBL10786998 0.81 KDM4E (0.38) LMNACYP3A4CYP2D6KDM4EALDH1A1
SCHEMBL7426725 0.79 LMNA (0.43) LMNATSPOKDM4EALDH1A1NPC1
SCHEMBL7435587 0.79 QPCT (0.38) LMNACYP3A4CYP2C19ALDH1A1GAA
SCHEMBL7446891 0.76 LMNA (0.41) LMNATSPOKDM4EALDH1A1NPC1
SCHEMBL7440283 0.73 KDR (0.44) LMNAKDM4EALDH1A1GAARAB9A
SCHEMBL7441183 0.72 LMNA (0.39) LMNATSPOKDM4EALDH1A1NPC1
SCHEMBL7447594 0.67 LCK (0.41) TSPOKDM4EALDH1A1NPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4880817-A O-functionalized derivatives of substituted isoquinolin-3-ols having cardiotonic and/or phosphodiesterase fraction III inhibiting properties and/or renal vasodilating properties ORTHO PHARMACEUTICAL CORPORATION (US) 1989-11-14 US claimed
US-4880817-A O-functionalized derivatives of substituted isoquinolin-3-ols having cardiotonic and/or phosphodiesterase fraction III inhibiting properties and/or renal vasodilating properties ORTHO PHARMACEUTICAL CORPORATION (US) 1989-11-14 US disclosed