SCHEMBL744078

SCHEMBL744078

O=C(/C=C\C(=O)ON(Br)c1ccccc1)ON(Br)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.40
TRPM8 Q7Z2W7 3/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HCAR2 Q8TDS4 3/20 0.38
ATM Q13315 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ALDH1A1 P00352 3/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
RAB9A P51151 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27324937 0.79 NPSR1 (0.43) NPSR1TRPM8MAPTKDM4EHPGD
SCHEMBL742918 0.76 NPSR1 (0.40) NPSR1TRPM8MAPTKDM4EHPGD
SCHEMBL11361015 0.76 NPSR1 (0.40) NPSR1TRPM8MAPTKDM4EHPGD
SCHEMBL28926817 0.72 HCAR2 (0.46) NPSR1TRPM8HCAR2TDP1ALDH1A1
SCHEMBL11055834 0.71 NPSR1 (0.35) NPSR1KDM4EATMTDP1L3MBTL1
SCHEMBL11205776 0.67 ALDH1A1 (0.34) NPSR1TRPM8MAPTKDM4EHPGD
SCHEMBL27636145 0.65 TDP1 (0.47) NPSR1MAPTKDM4EHPGDHSD17B10
SCHEMBL356193 0.64 HPGD (0.57) MAPTKDM4EHPGDHSD17B10HCAR2
SCHEMBL356194 0.64 HPGD (0.57) MAPTKDM4EHPGDHSD17B10HCAR2
SCHEMBL3042400 0.64 NPSR1 (0.50) NPSR1KDM4EATMTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431028-B1 FAST-DISSOLVING ORAL FILM FOR EFFECTIVELY CONCEALING UNPLEASANT TASTES CHABIO & DIOSTECH CO LTD (KR) 2017-07-12 EP claimed
US-9492379-B2 Quickly soluble oral film dosage containing steviosides as a unpleasant taste masking agent CHABIO & DIOSTECH CO., LTD. (KR) 2016-11-15 US claimed
US-20130039932-A1 QUICKLY SOLUBLE ORAL FILM DOSAGE CONTAINING STEVIOSIDES AS A UNPLEASANT TASTE MASKING AGENT CHABIO & DIOSTECH CO., LTD. (KR) 2013-02-14 US claimed
US-20120156229-A1 QUICKLY SOLUBLE ORAL FILM DOSAGE CONTAINING STEVIOSIDES AS A UNPLEASANT TASTE MASKING AGENT CHABIO & DIOSTECH CO. LTD (KR) 2012-06-21 US claimed
EP-2431028-A2 FAST-DISSOLVING ORAL FILM FOR EFFECTIVELY CONCEALING UNPLEASANT TASTES Chabio & Diostech Co., Ltd. (KR) 2012-03-21 EP claimed
EP-2431028-B1 FAST-DISSOLVING ORAL FILM FOR EFFECTIVELY CONCEALING UNPLEASANT TASTES CHABIO & DIOSTECH CO LTD (KR) 2017-07-12 EP disclosed
US-9492379-B2 Quickly soluble oral film dosage containing steviosides as a unpleasant taste masking agent CHABIO & DIOSTECH CO., LTD. (KR) 2016-11-15 US disclosed
US-20130039932-A1 QUICKLY SOLUBLE ORAL FILM DOSAGE CONTAINING STEVIOSIDES AS A UNPLEASANT TASTE MASKING AGENT CHABIO & DIOSTECH CO., LTD. (KR) 2013-02-14 US disclosed
US-20120156229-A1 QUICKLY SOLUBLE ORAL FILM DOSAGE CONTAINING STEVIOSIDES AS A UNPLEASANT TASTE MASKING AGENT CHABIO & DIOSTECH CO. LTD (KR) 2012-06-21 US disclosed
EP-2431028-A2 FAST-DISSOLVING ORAL FILM FOR EFFECTIVELY CONCEALING UNPLEASANT TASTES Chabio & Diostech Co., Ltd. (KR) 2012-03-21 EP disclosed
US-4847260-A NICOTINIC AND ISONITINIC ESTER ANTIARRHYTHMIA AGENTS FOR SKINS NITTO DENKO CORPORATION (JP) 1989-07-11 US disclosed
EP-0182635-B1 COMPOSITION FOR PERCUTANEOUS ADMINISTRATION NITTO DENKO CORPORATION (JP) 1989-05-31 EP disclosed
EP-0182635-A1 Composition for percutaneous administration NITTO DENKO CORPORATION (JP) 1986-05-28 EP disclosed