SCHEMBL7442115

SCHEMBL7442115

Sc1ccccc1C1=CCCC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
F2RL1 P55085 2/20 0.43
PTGS2 P35354 1/20 0.41
GRM2 Q14416 1/20 0.38
TDP1 Q9NUW8 1/20 0.35
IDO1 P14902 1/20 0.32
PSMB5 P28074 3/20 0.32
CCNE1 P24864 2/20 0.31
CDK2 P24941 2/20 0.31
CDK5 Q00535 1/20 0.31
KDR P35968 1/20 0.31
PDE10A Q9Y233 1/20 0.31
ACMSD Q8TDX5 1/20 0.31
CLCN2 P51788 1/20 0.31
ELANE P08246 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28758944 0.84 PTGS2 (0.51) F2RL1PTGS2GRM2TDP1PSMB5
SCHEMBL11815728 0.78 PTGS2 (0.59) F2RL1PTGS2GRM2TDP1PSMB5
SCHEMBL8784661 0.75 ALDH1A1 (0.48) F2RL1PTGS2GRM2TDP1IDO1
SCHEMBL2329786 0.75 PTGS2 (0.45) F2RL1PTGS2GRM2TDP1PSMB5
SCHEMBL27847334 0.75 PTGS2 (0.41) F2RL1PTGS2GRM2TDP1IDO1
SCHEMBL11824855 0.75 PTGS2 (0.45) F2RL1PTGS2GRM2TDP1PSMB5
SCHEMBL5863208 0.75 PTGS2 (0.41) F2RL1PTGS2GRM2TDP1IDO1
SCHEMBL6757109 0.75 F2RL1 (0.43) F2RL1PTGS2GRM2TDP1IDO1
SCHEMBL9806271 0.75 PTGS2 (0.57) F2RL1PTGS2GRM2ACMSDPPARA
SCHEMBL28618746 0.72 PTGS2 (0.46) F2RL1PTGS2GRM2TDP1PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5936128-A BENZENETHIOL COMPOUNDS AS INTERMEDIATES; BACTERICIDES, VIRICIDES; HIV WARNER-LAMBERT COMPANY (US) 1999-08-10 US claimed
US-5808062-A AIDS THERAPY WARNER-LAMBERT COMPANY (US) 1998-09-15 US claimed
EP-0729466-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP claimed
EP-0729463-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & COMPANY (US) 1996-09-04 EP claimed
WO-1995014011-A2 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO claimed
WO-1995014014-A2 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO claimed