SCHEMBL7442275

SCHEMBL7442275

O=C(c1ccc(NCCN2CCCC2)cc1-c1ccc(OCCN2CCCC2)cc1)c1csc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 12/20 0.47
ESR2 Q92731 11/20 0.47
F2 P00734 1/20 0.46
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
HSD17B10 Q99714 1/20 0.45
GCGR P47871 1/20 0.44
ITGA4 P13612 1/20 0.43
LTA4H P09960 2/20 0.42
MCHR1 Q99705 1/20 0.42
KDR P35968 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7451880 0.87 HRH3 (0.51) ESR1ESR2F2ALDH1A1CYP1A2
SCHEMBL7445232 0.85 ESR1 (0.57) ESR1ESR2ALDH1A1CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL8589966 0.84 ESR1 (0.58) ESR1ESR2ALDH1A1CYP1A2CYP2D6
SCHEMBL7414836 0.84 ESR1 (0.58) ESR1ESR2F2ALDH1A1CYP1A2
SCHEMBL7817318 0.84 ESR1 (0.48) ESR1ESR2F2ALDH1A1CYP1A2
SCHEMBL7444427 0.84 ESR1 (0.50) ESR1ESR2F2ALDH1A1CYP1A2
SCHEMBL7445743 0.84 ESR1 (0.59) ESR1ESR2F2ALDH1A1CYP1A2
SCHEMBL7452427 0.78 ESR1 (0.51) ESR1ESR2F2ALDH1A1CYP1A2
SCHEMBL7772092 0.77 ESR1 (0.56) ESR1ESR2F2ALDH1A1CYP1A2
SCHEMBL7442280 0.76 ESR1 (0.78) ESR1ESR2F2ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed