SCHEMBL7444427

SCHEMBL7444427

O=C(c1ccc(SCCN2CCCC2)cc1-c1ccc(OCCN2CCCC2)cc1)c1csc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 15/20 0.50
ESR2 Q92731 15/20 0.50
F2 P00734 1/20 0.48
ALDH1A1 P00352 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 2/20 0.46
HSD17B10 Q99714 2/20 0.46
CYP1A2 P05177 1/20 0.46
GCGR P47871 1/20 0.44
ITGA4 P13612 1/20 0.44
LTA4H P09960 1/20 0.43
MEN1 O00255 1/20 0.43
PLD2 O14939 1/20 0.43
KDM1A O60341 1/20 0.43
NR1I2 O75469 1/20 0.43
USP2 O75604 1/20 0.43
C5 P01031 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
FYN P06241 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7451880 0.88 HRH3 (0.51) ESR1ESR2F2ALDH1A1CYP2D6
SCHEMBL7445232 0.86 ESR1 (0.57) ESR1ESR2ALDH1A1CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL8589966 0.85 ESR1 (0.58) ESR1ESR2ALDH1A1CYP2D6CYP2C9
SCHEMBL7817318 0.85 ESR1 (0.48) ESR1ESR2F2ALDH1A1CYP2D6
SCHEMBL7414836 0.85 ESR1 (0.58) ESR1ESR2F2ALDH1A1CYP2D6
SCHEMBL7445743 0.84 ESR1 (0.59) ESR1ESR2F2ALDH1A1CYP2D6
SCHEMBL7442275 0.84 ESR1 (0.47) ESR1ESR2F2ALDH1A1CYP2D6
SCHEMBL7772092 0.78 ESR1 (0.56) ESR1ESR2F2ALDH1A1CYP2D6
SCHEMBL6597254 0.77 ESR1 (0.79) ESR1ESR2F2ALDH1A1CYP2D6
SCHEMBL7452427 0.77 ESR1 (0.51) ESR1ESR2F2ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed