SCHEMBL7442897

SCHEMBL7442897

CN(C)CCOc1ccc(-c2cccc(O)c2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.69
CHRNA4 P43681 1/20 0.69
KDR P35968 6/20 0.58
LSS P48449 1/20 0.58
HSD17B1 P14061 2/20 0.52
HSD17B2 P37059 2/20 0.52
CYP3A4 P08684 2/20 0.52
CYP2C9 P11712 1/20 0.52
LTA4H P09960 2/20 0.51
KEAP1 Q14145 1/20 0.51
NFE2L2 Q16236 1/20 0.51
ESR1 P03372 6/20 0.49
HRH3 Q9Y5N1 1/20 0.49
ESR2 Q92731 3/20 0.48
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5141140 0.85 KDR (0.67) CHRNB2CHRNA4KDRHSD17B1HSD17B2
SCHEMBL8264173 0.83 LSS (0.59) CHRNB2CHRNA4LSSLTA4HKEAP1
SCHEMBL29591093 0.82 CHRNB2 (1.00) CHRNB2CHRNA4LTA4HKEAP1NFE2L2
SCHEMBL1957431 0.82 CHRNB2 (1.00) CHRNB2CHRNA4LTA4HKEAP1NFE2L2
SCHEMBL7346114 0.82 HSD17B1 (0.61) KDRHSD17B1HSD17B2CYP3A4CYP2C9
SCHEMBL22831331 0.82 LSS (0.83) LSSCYP3A4LTA4HKEAP1NFE2L2
SCHEMBL24721056 0.81 LSS (0.56) CHRNB2CHRNA4LSSCYP3A4LTA4H
SCHEMBL30956050 0.80 HSD17B1 (0.53) KDRLSSHSD17B1HSD17B2CYP3A4
SCHEMBL30387666 0.80 HSD17B1 (0.57) KDRLSSHSD17B1HSD17B2CYP3A4
SCHEMBL24721332 0.79 LSS (0.55) CHRNB2CHRNA4LSSLTA4HKEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed