SCHEMBL8264173

SCHEMBL8264173

Cc1cccc(-c2ccc(OCCN(C)C)cc2)c1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LSS P48449 1/20 0.59
ESR1 P03372 2/20 0.57
ESR2 Q92731 1/20 0.57
LTA4H P09960 2/20 0.53
KEAP1 Q14145 1/20 0.53
NFE2L2 Q16236 1/20 0.53
ACHE P22303 2/20 0.52
TNKS O95271 2/20 0.50
HRH3 Q9Y5N1 1/20 0.50
CHRNB2 P17787 1/20 0.50
CHRNA4 P43681 1/20 0.50
HCRTR1 O43613 1/20 0.47
MAOB P27338 1/20 0.47
ITGA4 P13612 1/20 0.46
NAPEPLD Q6IQ20 1/20 0.46
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8264198 0.92 LSS (0.71) LSSESR1ESR2ACHEHRH3
SCHEMBL8264812 0.89 CHRNB2 (0.59) ESR1ESR2LTA4HKEAP1NFE2L2
SCHEMBL22831331 0.83 LSS (0.83) LSSESR1ESR2LTA4HKEAP1
SCHEMBL7442897 0.83 CHRNB2 (0.69) LSSESR1ESR2LTA4HKEAP1
SCHEMBL8264152 0.82 FFAR4 (0.50) LSSALDH1A1
SCHEMBL8265107 0.82 CYP3A4 (0.47) LSSLTA4HCHRNB2CHRNA4ALDH1A1
SCHEMBL24721056 0.82 LSS (0.56) LSSESR1ESR2LTA4HKEAP1
SCHEMBL8360713 0.82 CHRNB2 (0.67) ESR1LTA4HKEAP1NFE2L2CHRNB2
SCHEMBL8264819 0.81 MAOB (0.58) LSSESR1CHRNB2CHRNA4MAOB
SCHEMBL8264189 0.81 TAAR1 (0.48) LSSLTA4HMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2177518-A1 Organic compounds Novartis AG (CH) 2010-04-21 EP disclosed
EP-1833816-B1 SUBSTITUTED PIPERIDINES AS RENIN INHIBITORS NOVARTIS AG (CH) 2009-11-11 EP disclosed
WO-2006069788-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2006-07-06 WO disclosed