SCHEMBL7443013

SCHEMBL7443013

O=C(O)c1cc2c([nH]1)C(=O)C=CC2=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.48
NFKB1 P19838 1/20 0.48
BLM P54132 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
ALDH1A1 P00352 2/20 0.44
LMNA P02545 1/20 0.44
CYP2C19 P33261 2/20 0.41
GPR35 Q9HC97 4/20 0.41
TSHR P16473 1/20 0.39
IDO1 P14902 1/20 0.38
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 2/20 0.37
MEN1 O00255 1/20 0.37
GRIN2D O15399 1/20 0.37
GRIN3B O60391 1/20 0.37
CYP1A2 P05177 1/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12390669 0.68 IDO1 (0.41) SMN1; SMN2ALDH1A1IDO1KDM4EGRIN2D
SCHEMBL7816527 0.68 GAA (0.41) SMN1; SMN2ALDH1A1LMNACYP2C19TSHR
SCHEMBL6513260 0.67 KDM4E (0.49) ALOX15NFKB1BLMSMN1; SMN2ALDH1A1
SCHEMBL1259832 0.67 HSD17B10 (0.47) ALOX15NFKB1BLMSMN1; SMN2ALDH1A1
Chelidamic Acid SCHEMBL742928 0.66 ALOX15 (1.00) ALOX15NFKB1BLMSMN1; SMN2ALDH1A1
SCHEMBL7830760 0.64 ALDH1A1 (0.44) SMN1; SMN2ALDH1A1IDO1KDM4EHPGD
Chelidamic Acid SCHEMBL9658074 0.64 ALOX15 (0.95) ALOX15NFKB1BLMSMN1; SMN2ALDH1A1
Chelidamic Acid SCHEMBL1176783 0.64 ALOX15 (0.95) ALOX15NFKB1BLMSMN1; SMN2ALDH1A1
SCHEMBL1006834 0.64 ALOX15 (0.48) ALOX15NFKB1BLMSMN1; SMN2ALDH1A1
SCHEMBL27960983 0.64 KDM4E (0.37) ALDH1A1CYP2C19IDO1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706525-A1 ANTIHYPERTENSIVE TRICYCLIC AZEPINE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE Novartis AG (CH) 1996-04-17 EP disclosed
WO-1995001353-A1 ANTIHYPERTENSIVE TRICYCLIC AZEPINE DERIVATIVES USEFUL AS INHIBITORS OF ENKEPHALINASE AND ACE CIBA-GEIGY AG (CH) 1995-01-12 WO disclosed