SCHEMBL7443167

SCHEMBL7443167

Cc1cc(Nc2ccc(-c3ccccc3C(=O)O)cc2)n2nccc2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.50
ALDH1A1 P00352 4/20 0.50
MAPT P10636 4/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
LMNA P02545 3/20 0.50
NPC1 O15118 2/20 0.50
HPGD P15428 2/20 0.50
RAB9A P51151 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
CLK1 P49759 1/20 0.50
RXFP1 Q9HBX9 1/20 0.44
MAPK1 P28482 3/20 0.44
HTT P42858 1/20 0.44
GAA P10253 1/20 0.43
ATM Q13315 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
OPRL1 P41146 1/20 0.40
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7437229 0.87 PRKAB2 (0.44) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL7448477 0.82 FNTA (0.42) KDM4EALDH1A1OPRL1USP2TSHR
SCHEMBL7434502 0.82 MEN1 (0.45) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL7443760 0.82 MEN1 (0.45) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL8555494 0.82 HPGD (0.51) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL7435550 0.77 BCL6 (0.42) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL7440794 0.76 MEN1 (0.39) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL8554435 0.73 ALDH1A1 (0.67) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL7442147 0.73 FNTA (0.41)
SCHEMBL14427338 0.70 CDK2 (0.57) ALDH1A1MEN1KMT2AMAPK1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed