SCHEMBL8554435

SCHEMBL8554435

COC(=O)c1ccccc1Nc1cc(C)nc2ccnn12

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.67
HPGD P15428 3/20 0.67
TP53 P04637 1/20 0.54
KDM4E B2RXH2 7/20 0.53
MAPT P10636 3/20 0.53
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ALOX15 P16050 1/20 0.49
POLB P06746 2/20 0.48
LMNA P02545 2/20 0.48
HSD17B10 Q99714 3/20 0.46
ATM Q13315 1/20 0.46
GLA P06280 2/20 0.44
GFER P55789 1/20 0.43
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555494 0.88 HPGD (0.51) ALDH1A1HPGDTP53KDM4EMAPT
SCHEMBL351286 0.76 F2 (0.40) ALDH1A1HPGDKDM4EMAPTKMT2A
SCHEMBL27728859 0.75 ALDH1A1 (0.65) ALDH1A1HPGDTP53KDM4EMAPT
Hydrochloric Acid SCHEMBL27749316 0.74 ALDH1A1 (0.63) ALDH1A1HPGDTP53KDM4EMAPT
SCHEMBL7443167 0.73 KDM4E (0.50) ALDH1A1HPGDKDM4EMAPTKMT2A
SCHEMBL1819140 0.72 GFER (0.71) ALDH1A1HPGDMAPTKMT2AMEN1
SCHEMBL1815233 0.71 HPGD (0.58) ALDH1A1HPGDTP53KDM4EMAPT
SCHEMBL22862844 0.70 KCNN3 (0.51) ALDH1A1HPGDKDM4EMAPTKMT2A
SCHEMBL13730760 0.70 ALDH1A1 (0.63) ALDH1A1HPGDKDM4EMAPTKMT2A
SCHEMBL19065779 0.70 MAPT (0.79) ALDH1A1HPGDKDM4EMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0591528-B1 PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVE AND ANTI-INFLAMMATORY CONTAINING THE SAME OTSUKA PHARMA CO LTD (JP) 1998-12-23 EP disclosed
US-5688949-A CYCLOOXYGENASE INHIBITORS OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1997-11-18 US disclosed
EP-0591528-A1 PYRAZOLO 1,5-a]PYRIMIDINE DERIVATIVE AND ANTI-INFLAMMATORY CONTAINING THE SAME OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1994-04-13 EP disclosed