SCHEMBL7443174

SCHEMBL7443174

O=C(c1ccc(OCCN2CCCCC2)cc1)c1ccccc1-c1ccc(OCCN2CCCC2)cc1

nearest known ligand 0.70

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PSMB1 P20618 3/20 0.70
PSMB5 P28074 3/20 0.70
PSMB2 P49721 2/20 0.70
LTA4H P09960 2/20 0.69
GCGR P47871 2/20 0.68
KCNH2 Q12809 1/20 0.67
HRH3 Q9Y5N1 1/20 0.67
KDM4E B2RXH2 3/20 0.60
ALDH1A1 P00352 2/20 0.60
DRD2 P14416 1/20 0.59
DRD1 P21728 1/20 0.59
DRD3 P35462 1/20 0.59
HRH4 Q9H3N8 1/20 0.58
ESR1 P03372 7/20 0.57
ESR2 Q92731 6/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7445638 0.99 LTA4H (0.70) PSMB1PSMB5PSMB2LTA4HGCGR
SCHEMBL7352552 0.94 LTA4H (0.65) PSMB1PSMB5PSMB2LTA4HGCGR
SCHEMBL7439685 0.93 LTA4H (0.63) PSMB1PSMB5PSMB2LTA4HGCGR
SCHEMBL8711348 0.85 LTA4H (0.76) PSMB1PSMB5PSMB2LTA4HGCGR
SCHEMBL7748549 0.85 ESR1 (0.66) PSMB1PSMB5PSMB2LTA4HGCGR
SCHEMBL3092657 0.84 ESR1 (0.65) PSMB1PSMB5PSMB2KCNH2ALDH1A1
SCHEMBL13305534 0.83 LTA4H (0.97) PSMB1PSMB5PSMB2LTA4HGCGR
SCHEMBL8599886 0.83 ESR1 (0.65) PSMB1PSMB5PSMB2LTA4HGCGR
SCHEMBL7738182 0.83 ESR1 (0.64) PSMB1PSMB5PSMB2LTA4HKCNH2
SCHEMBL8588964 0.82 LTA4H (0.64) PSMB1PSMB5PSMB2LTA4HGCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed