SCHEMBL8711348

SCHEMBL8711348

O=C(O)c1ccccc1C(=O)c1ccc(OCCN2CCCCC2)cc1

nearest known ligand 0.76

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.76
PSMB1 P20618 4/20 0.73
PSMB5 P28074 4/20 0.73
PSMB2 P49721 3/20 0.73
GCGR P47871 2/20 0.71
KDM4E B2RXH2 4/20 0.66
ALDH1A1 P00352 2/20 0.66
DRD2 P14416 1/20 0.65
DRD1 P21728 1/20 0.65
DRD3 P35462 1/20 0.65
HRH4 Q9H3N8 1/20 0.64
ESR1 P03372 3/20 0.60
ESR2 Q92731 2/20 0.59
HTT P42858 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13305534 0.88 LTA4H (0.97) LTA4HPSMB1PSMB5PSMB2GCGR
SCHEMBL8711352 0.88 LTA4H (0.69) LTA4HPSMB1PSMB5PSMB2GCGR
Pitofenone SCHEMBL2111794 0.87 KDM4E (0.69) LTA4HPSMB1PSMB5PSMB2GCGR
SCHEMBL28380360 0.87 LTA4H (1.00) LTA4HPSMB1PSMB5PSMB2GCGR
Pitofenone SCHEMBL4389235 0.86 KDM4E (0.67) LTA4HPSMB1PSMB5PSMB2GCGR
SCHEMBL7443174 0.85 PSMB1 (0.70) LTA4HPSMB1PSMB5PSMB2GCGR
SCHEMBL7445638 0.84 LTA4H (0.70) LTA4HPSMB1PSMB5PSMB2GCGR
SCHEMBL8714269 0.84 PSMB1 (0.64) LTA4HPSMB1PSMB5PSMB2GCGR
Hydrochloric Acid SCHEMBL9191319 0.84 PSMB1 (0.64) LTA4HPSMB1PSMB5PSMB2GCGR
SCHEMBL2741667 0.84 PSMB1 (0.80) LTA4HPSMB1PSMB5PSMB2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0364941-B1 Branched-chain alkyl esters of 2-(4-(2-piperidino ethoxy)benzoyl)benzoic acid, processes for their preparation and their use as spasmolytic agents HOECHST AG (DE) 1995-02-15 EP claimed
JP-2169585-A None JP disclosed
US-5821252-A PROLONGED SPASMOLYTIC AND ANESTHETIC ACITIVITY HOECHST AKTIENGESELLSCHAFT (DE) 1998-10-13 US disclosed
EP-0364941-B1 Branched-chain alkyl esters of 2-(4-(2-piperidino ethoxy)benzoyl)benzoic acid, processes for their preparation and their use as spasmolytic agents HOECHST AG (DE) 1995-02-15 EP disclosed
EP-0364941-B1 Branched-chain alkyl esters of 2-(4-(2-piperidino ethoxy)benzoyl)benzoic acid, processes for their preparation and their use as spasmolytic agents HOECHST AG (DE) 1995-02-15 EP disclosed
CN-1025615-C Branched-chain alkyl esters of 2-[4-(2-piperidiono-ethoxy)-benzoyl]-benzoic acid, processes for their preparation and their use as spasmolytic agents HOECHST AG (DE) 1994-08-10 CN disclosed
CN-1025615-C Branched-chain alkyl esters of 2-[4-(2-piperidiono-ethoxy)-benzoyl]-benzoic acid, processes for their preparation and their use as spasmolytic agents HOECHST AG (DE) 1994-08-10 CN disclosed
JP-H02169585-A BRANCHED CHAIN ALKYL ESTER OF 2-(4-(2-PIPERIDINO-ETHOXY)-BENZOYL)BENZOATE AND ITS PRODUCTION HOECHST AG 1990-06-29 JP disclosed
EP-0364941-A1 Branched-chain alkyl esters of 2-(4-(2-piperidino ethoxy)benzoyl)benzoic acid, processes for their preparation and their use as spasmolytic agents HOECHST AKTIENGESELLSCHAFT (DE) 1990-04-25 EP disclosed
EP-0364941-A1 Branched-chain alkyl esters of 2-(4-(2-piperidino ethoxy)benzoyl)benzoic acid, processes for their preparation and their use as spasmolytic agents HOECHST AKTIENGESELLSCHAFT (DE) 1990-04-25 EP disclosed