SCHEMBL7444076

SCHEMBL7444076

NN=Cc1ccc(CNC(=O)c2ccc3c(c2)CN(CCC(=O)O)C(=O)CC3)cc1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.48
ITGA2B P08514 5/20 0.48
ITGA2 P17301 2/20 0.43
NAMPT P43490 6/20 0.41
ROCK2 O75116 1/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
PPARG P37231 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPK14 Q16539 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7444067 0.85 ITGB3 (0.65) ITGB3ITGA2BITGA2NAMPT
SCHEMBL6677682 0.73 ITGB3 (0.54) ITGB3ITGA2BALDH1A1
SCHEMBL7396984 0.73 ITGB3 (0.75) ITGB3ITGA2BITGA2HDAC1HDAC8
SCHEMBL7442215 0.71 ITGB3 (0.63) ITGB3ITGA2B
SCHEMBL6678690 0.70 ITGB3 (0.53) ITGB3ITGA2BNAMPT
SCHEMBL6676580 0.70 ITGB3 (0.48) ITGB3ITGA2BNAMPTALDH1A1
Trifluoroacetic Acid SCHEMBL8182682 0.69 ITGB3 (0.68) ITGB3ITGA2BITGA2HDAC1HDAC8
Hydrochloric Acid SCHEMBL7659033 0.69 ITGB3 (0.54) ITGB3ITGA2BALDH1A1
SCHEMBL7373451 0.67 PPARG (0.65) ITGB3ITGA2BHDAC8HDAC6PPARG
SCHEMBL7444173 0.67 ITGB3 (0.72) ITGB3ITGA2BITGA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403578-B1 ANTICOAGULANTS, CARDIOVASCULAR DISORDERS SMITHKLINE BEECHAM CORPORATION 2002-06-11 US disclosed
EP-0674623-A1 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1995-10-04 EP disclosed
WO-1994014776-A2 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1994-07-07 WO disclosed