SCHEMBL7444093

SCHEMBL7444093

Cc1cc(C(=O)c2ccsc2)ccc1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.47
DYRK1B Q9Y463 1/20 0.47
HSD17B1 P14061 7/20 0.47
HSD17B2 P37059 7/20 0.47
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
LCK P06239 1/20 0.44
FYN P06241 1/20 0.44
DAO P14920 1/20 0.44
SLC22A6 Q4U2R8 1/20 0.42
SLC22A8 Q8TCC7 1/20 0.42
HDAC1 Q13547 1/20 0.41
SIRT1 Q96EB6 1/20 0.39
HSD17B14 Q9BPX1 1/20 0.39
TP53 P04637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PDK1 Q15118 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31621156 0.84 HTT (0.61) DYRK1ADYRK1BHSD17B1HSD17B2HTT
SCHEMBL1758239 0.84 HTT (0.61) DYRK1ADYRK1BHSD17B1HSD17B2HTT
SCHEMBL6961496 0.82 KMT2A (0.47) HTTSMN1; SMN2CES2CES1LCK
SCHEMBL11053174 0.82 HTT (0.64) DYRK1ADYRK1BHSD17B1HSD17B2HTT
SCHEMBL31574429 0.80 HTT (0.57) DYRK1ADYRK1BHSD17B1HSD17B2HTT
SCHEMBL7444751 0.80 CYP1A2 (0.53) HTTCES2CES1SLC22A6SLC22A8
SCHEMBL6958930 0.80 SLC22A6 (0.73) HSD17B2HTTSLC22A6SLC22A8POLB
SCHEMBL6961510 0.78 KDM4E (0.43) HTTSMN1; SMN2CES2CES1LCK
SCHEMBL2166098 0.78 CES2 (0.71) HTTCES2CES1LCKFYN
SCHEMBL1758781 0.77 HTT (0.75) DYRK1ADYRK1BHSD17B1HSD17B2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed