SCHEMBL7444174

SCHEMBL7444174

O=C(c1ccc(F)cc1)[C@H]1CC[C@H]2CN(CCc3ccccc3)CCN2C1

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.59
HTR2C P28335 4/20 0.59
HTR7 P34969 4/20 0.59
HTR6 P50406 4/20 0.59
KDM4E B2RXH2 2/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
SLC18A3 Q16572 2/20 0.50
MEN1 O00255 1/20 0.50
MAPK1 P28482 1/20 0.50
KMT2A Q03164 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7444169 1.00 HTR2A (0.59) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL7444179 1.00 HTR2A (0.59) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL8642581 0.89 SLC18A3 (0.62) HTR2AHTR2CKDM4ECYP1A2CYP3A4
SCHEMBL1582470 0.81 HTR2A (0.87) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL8646880 0.81 KDM2B (0.53) HTR2AHTR2CHTR7HTR6
SCHEMBL467405 0.81 KDM2B (0.53) HTR2AHTR2CHTR7HTR6
SCHEMBL467403 0.81 KDM2B (0.53) HTR2AHTR2CHTR7HTR6
SCHEMBL467404 0.81 KDM2B (0.53) HTR2AHTR2CHTR7HTR6
Hydrochloric Acid SCHEMBL7418228 0.80 HTR2A (0.85) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL8641073 0.77 HTR2A (0.58) HTR2AHTR2CHTR7HTR6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731307-A Neuroleptic 2,7-disubtituted perhydro-1h-pyrido 1, 2-A!pyrazines PFIZER, INC. (US) 1998-03-24 US claimed
WO-1996010570-A1 NEUROLEPTIC 2,7-DISUBSTITUTED PERHYDRO-1H-PYRIDO[1,2-a]PYRAZINES PFIZER INC. (US) 1996-04-11 WO claimed