SCHEMBL8641073

SCHEMBL8641073

OC(c1ccc(F)cc1)[C@H]1CC[C@H]2CN(CCc3ccccc3)CCN2C1

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.58
HTR2C P28335 3/20 0.58
HTR7 P34969 2/20 0.58
KDM4E B2RXH2 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
TSHR P16473 1/20 0.54
HTR6 P50406 1/20 0.48
SLC6A4 P31645 1/20 0.48
SLC6A3 Q01959 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433902 0.83 HTR2A (0.47) HTR2AHTR2CHTR7SLC6A4SLC6A3
SCHEMBL8645119 0.83 HTR2A (0.47) HTR2AHTR2CHTR7SLC6A4SLC6A3
SCHEMBL8642030 0.81 HTR2A (0.45) HTR2AHTR2CHTR7CYP2D6HTR6
SCHEMBL9330147 0.81 HTR2A (0.87) HTR2AHTR2CHTR7KDM4ECYP1A2
SCHEMBL7444174 0.77 HTR2A (0.59) HTR2AHTR2CHTR7KDM4ECYP1A2
SCHEMBL7444179 0.77 HTR2A (0.59) HTR2AHTR2CHTR7KDM4ECYP1A2
SCHEMBL7444169 0.77 HTR2A (0.59) HTR2AHTR2CHTR7KDM4ECYP1A2
SCHEMBL9328582 0.76 HTR2A (0.87) HTR2AHTR2CHTR7KDM4ECYP1A2
SCHEMBL8643172 0.73 SIGMAR1 (0.47)
SCHEMBL9375973 0.73 HTR2A (1.00) HTR2AHTR2CHTR7KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731307-A Neuroleptic 2,7-disubtituted perhydro-1h-pyrido 1, 2-A!pyrazines PFIZER, INC. (US) 1998-03-24 US claimed