SCHEMBL7444528

SCHEMBL7444528

Cc1ccc2[nH]c(-c3cccc(C(=O)O)c3)nc2c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.71
ALDH1A1 P00352 5/20 0.71
HPGD P15428 4/20 0.71
NPC1 O15118 4/20 0.71
RAB9A P51151 4/20 0.71
SMN1; SMN2 Q16637 3/20 0.71
MMP2 P08253 5/20 0.54
MMP9 P14780 5/20 0.54
MMP8 P22894 5/20 0.54
PIN1 Q13526 1/20 0.51
MMP13 P45452 3/20 0.50
MAPT P10636 2/20 0.50
PPARG P37231 1/20 0.50
PPARA Q07869 1/20 0.50
COMT P21964 1/20 0.50
TP53 P04637 1/20 0.50
PKM P14618 1/20 0.50
GFER P55789 1/20 0.50
KMT2A Q03164 5/20 0.49
FHIT P49789 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31412081 0.89 KDM4E (0.79) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL11599505 0.88 KDM4E (0.77) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL15249611 0.86 ALDH1A1 (0.67) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL28640195 0.85 KDM4E (0.73) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL7943525 0.85 KDM4E (0.63) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL31533522 0.85 KDM4E (0.72) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL6124304 0.84 NPC1 (0.61) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL1806763 0.84 KDM4E (0.71) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL31679082 0.83 KDM4E (1.00) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL4714012 0.83 KDM4E (1.00) KDM4EALDH1A1HPGDNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968191-A1 PHENYLBENZIMIDAZOLE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2000-01-05 EP disclosed
WO-1998034923-A1 PHENYLBENZIMIDAZOLE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 1998-08-13 WO disclosed