SCHEMBL7444560

SCHEMBL7444560

O=C(N1CCNCC1)N1CCN(c2ccncc2)CC1

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.66
NCF1 P14598 1/20 0.66
PLD1 Q13393 1/20 0.66
AKR1C3 P42330 6/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
TRPV1 Q8NER1 1/20 0.49
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 1/20 0.47
CHKA P35790 2/20 0.47
ALDH1A1 P00352 3/20 0.47
GAA P10253 1/20 0.47
CYP3A4 P08684 1/20 0.47
TSHR P16473 1/20 0.47
LMNA P02545 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
ITGB3 P05106 2/20 0.46
ITGA2B P08514 2/20 0.46
CA2 P00918 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16599286 0.90 AKR1C3 (0.58) AKR1C3SMN1; SMN2TRPV1CYP2C9CYP2C19
SCHEMBL8838202 0.83 AKR1C3 (0.54) AKR1C3SMN1; SMN2TRPV1CYP2C9CYP2C19
SCHEMBL27471218 0.83 ALDH1A1 (0.66) AKR1C3SMN1; SMN2TRPV1CYP2C9CYP2C19
SCHEMBL6180189 0.81 ALDH1A1 (0.58) ADRB2NCF1PLD1SMN1; SMN2CYP2C9
SCHEMBL894239 0.80 ADRB2 (1.00) ADRB2NCF1PLD1CYP2C9CYP2C19
SCHEMBL74335 0.80 ADRB2 (1.00) ADRB2NCF1PLD1CYP2C9CYP2C19
Acetic Acid SCHEMBL27482977 0.80 ADRB2 (0.76) ADRB2NCF1PLD1CYP2C9CYP2C19
Formaldehyde SCHEMBL28065716 0.79 ADRB2 (0.88) ADRB2NCF1PLD1CYP2C9CYP2C19
SCHEMBL6179989 0.79 LSS (0.59) ADRB2NCF1PLD1ITGB3ITGA2B
SCHEMBL6791781 0.79 ITGB3 (0.57) ADRB2NCF1PLD1ALDH1A1ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6440972-B1 Heterocyclic compounds useful as oxido-squalene cyclase inhibitors ZENECA LIMITED (GB) 2002-08-27 US disclosed
EP-0966460-A1 HETEROCYCLIC COMPOUNDS USEFUL AS OXIDO-SQUALENE CYCLASE INHIBITORS ZENECA LIMITED (GB) 1999-12-29 EP disclosed
WO-1998035956-A1 HETEROCYCLIC COMPOUNDS USEFUL AS OXIDO-SQUALENE CYCLASE INHIBITORS ZENECA LIMITED (US) 1998-08-20 WO disclosed