SCHEMBL7444669

SCHEMBL7444669

Cc1ccc2[nH]c(-c3cccc(CN4CCOCC4)c3)nc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.57
KIT P10721 3/20 0.55
CNR1 P21554 3/20 0.51
CNR2 P34972 3/20 0.51
FGFR1 P11362 1/20 0.49
FGFR2 P21802 1/20 0.49
FGFR3 P22607 1/20 0.49
KDR P35968 1/20 0.49
ACHE P22303 1/20 0.49
AURKA O14965 1/20 0.47
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
HSD17B10 Q99714 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
GRIN2B Q13224 2/20 0.46
PSMB8 P28062 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC8 Q9BY41 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18237008 0.81 HDAC6 (0.68) PARP1KITCNR1CNR2AURKA
SCHEMBL6124304 0.77 NPC1 (0.61) ALDH1A1HPGDHSD17B10
SCHEMBL7449604 0.77 ATR (0.58) FGFR1KDRALDH1A1HPGDL3MBTL1
SCHEMBL1665040 0.76 PARP1 (0.53) PARP1AURKAALDH1A1HPGDHSD17B10
SCHEMBL24061140 0.76 HRH3 (0.58) CNR1CNR2ALDH1A1HPGDPSMB8
SCHEMBL21087331 0.75 NPC1 (0.60) KDRALDH1A1HPGDHSD17B10
SCHEMBL8262963 0.75 FGFR1 (0.51) PARP1FGFR1FGFR2FGFR3KDR
SCHEMBL18229495 0.75 HDAC6 (0.79) PARP1ACHEAURKAHDAC3HDAC1
SCHEMBL178443 0.74 NCF1 (0.66) ALDH1A1HPGDNCF1
SCHEMBL31478684 0.73 CNR2 (0.55) PARP1KITCNR1CNR2AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968191-A1 PHENYLBENZIMIDAZOLE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2000-01-05 EP claimed
WO-1998034923-A1 PHENYLBENZIMIDAZOLE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 1998-08-13 WO claimed