SCHEMBL7445138

SCHEMBL7445138

CCCCOC(=O)[C@@](N)(CC(=O)O)c1ccc(O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.49
ESR1 P03372 4/20 0.49
CYP1A2 P05177 3/20 0.49
MAPK1 P28482 2/20 0.49
LMNA P02545 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP2D6 P10635 1/20 0.49
NR1H2 P55055 1/20 0.49
RNASEL Q05823 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CHRM2 P08172 3/20 0.42
CHRM1 P11229 2/20 0.41
CHRM4 P08173 1/20 0.41
CHRM3 P20309 1/20 0.41
ALDH1A1 P00352 4/20 0.41
TDP1 Q9NUW8 3/20 0.41
CYP3A4 P08684 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
S1PR4 O95977 1/20 0.40
S1PR1 P21453 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5262276 0.80 S1PR1 (0.37) TSHRESR1CYP1A2MAPK1LMNA
SCHEMBL3525214 0.77 ESR1 (0.44) TSHRESR1CYP1A2MAPK1LMNA
SCHEMBL3654422 0.77 TSHR (0.50) TSHRESR1CYP1A2MAPK1LMNA
SCHEMBL4496293 0.75 TSHR (0.51) TSHRESR1CYP1A2MAPK1LMNA
SCHEMBL28264509 0.74 ESR1 (0.54) TSHRESR1CYP1A2MAPK1LMNA
SCHEMBL27315973 0.74 PIN1 (0.47) TSHRCYP2C19SMN1; SMN2CHRM2CHRM1
SCHEMBL12708518 0.72 ESR1 (0.48) TSHRESR1CYP1A2MAPK1LMNA
SCHEMBL30309035 0.71 ALDH1A1 (0.44) TSHRESR1CYP1A2MAPK1LMNA
SCHEMBL28137293 0.71 TSHR (0.51) TSHRCYP1A2MAPK1LMNACYP2C19
SCHEMBL27596964 0.70 ALDH1A1 (0.42) TSHRCYP1A2MAPK1LMNACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1034164-A4 SUBSTITUTED BETA-ALANINE DERIVATIVES AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2001-07-11 EP disclosed
EP-1034164-A1 SUBSTITUTED BETA-ALANINE DERIVATIVES AS CELL ADHESION INHIBITORS Merck & Co., Inc. (US) 2000-09-13 EP disclosed
WO-1999026921-A1 SUBSTITUTED β-ALANINE DERIVATIVES AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-06-03 WO disclosed