SCHEMBL7445375

SCHEMBL7445375

O=C1OC(CCc2ccc3c(c2)OCO3)(c2ccccc2)CC(O)=C1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CALM1 P0DP23 2/20 0.43
TRPM8 Q7Z2W7 1/20 0.42
HPGD P15428 3/20 0.42
ALDH1A1 P00352 3/20 0.42
MAPK1 P28482 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HDAC1 Q13547 2/20 0.41
RAB9A P51151 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
NPC1 O15118 1/20 0.41
LMNA P02545 2/20 0.40
EDNRB P24530 1/20 0.40
EDNRA P25101 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6602959 0.84 LDHA (0.41) GAA
SCHEMBL6605273 0.84 HPGD (0.44) CALM1TRPM8HPGDALDH1A1MAPK1
SCHEMBL6604225 0.82 CALM1 (0.43) CALM1TRPM8HPGDALDH1A1MAPK1
SCHEMBL6604754 0.82 HPGD (0.42) CALM1HPGDALDH1A1RAB9ANPC1
SCHEMBL7445786 0.75 ALDH1A1 (0.39) HPGDALDH1A1MAPK1KDM4EGLA
SCHEMBL6605035 0.72 LDHA (0.42)
SCHEMBL6604273 0.71 LDHA (0.39) ALDH1A1KDM4EHDAC1HDAC3HDAC2
SCHEMBL6608872 0.69 LDHA (0.41) KDM4EGAALMNAMEN1KMT2A
SCHEMBL6609678 0.69 LDHA (0.40) MAPK1KDM4EGAAEDNRBEDNRA
SCHEMBL6607939 0.68 LDHA (0.50) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729463-B1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & CO (US) 2002-05-22 EP claimed
WO-1995014011-A2 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO claimed