SCHEMBL7445475

SCHEMBL7445475

Cc1cc(NCc2ccc(-n3cccc3-c3nnn[nH]3)cc2)n2nccc2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN3 Q9UGI6 7/20 0.41
KCNN1 Q92952 1/20 0.41
KCNN2 Q9H2S1 1/20 0.41
CDK2 P24941 4/20 0.38
GAA P10253 1/20 0.37
PDE10A Q9Y233 2/20 0.37
CCNE1 P24864 3/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
GPR39 O43194 1/20 0.35
AGTR1 P30556 1/20 0.35
BRD4 O60885 1/20 0.35
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA2 P54646 1/20 0.35
PRKAA1 Q13131 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7440140 0.89 PRKAB2 (0.48) KCNN3KCNN1KCNN2CDK2PDE10A
SCHEMBL7440104 0.84 KMT2A (0.43) CDK2GAAMEN1NPC1RAB9A
SCHEMBL7449376 0.84 SMN1; SMN2 (0.37) GAAMEN1NPC1RAB9AKMT2A
SCHEMBL7438553 0.83 BRD4 (0.36) TP53MAPTBRD4
SCHEMBL7439844 0.83 KCNN3 (0.39) KCNN3KCNN1KCNN2CDK2GAA
SCHEMBL7438720 0.80 KCNN3 (0.47) KCNN3KCNN1KCNN2CDK2GAA
SCHEMBL7440798 0.80 AGTR1 (0.32) GAAMEN1NPC1RAB9AKMT2A
SCHEMBL7449569 0.79 KCNN3 (0.42) KCNN3KCNN1KCNN2CDK2GAA
SCHEMBL7445460 0.79 DPP4 (0.39)
SCHEMBL7435614 0.78 GSK3B (0.42) CDK2CCNE1MEN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed