SCHEMBL7445604

SCHEMBL7445604

N#Cc1ccccc1-c1ccc(CNc2cc(Cl)nc3ccnn23)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN3 Q9UGI6 14/20 0.66
KCNN1 Q92952 2/20 0.66
KCNN2 Q9H2S1 2/20 0.66
PDE10A Q9Y233 1/20 0.47
CDK2 P24941 3/20 0.45
CCNE1 P24864 2/20 0.44
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
BLM P54132 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7437667 0.88 PRKAB2 (0.51) KCNN3KCNN1KCNN2CDK2CCNE1
SCHEMBL7441417 0.88 MEN1 (0.49) KCNN3KCNN1KCNN2CDK2CCNE1
SCHEMBL7435705 0.84 KCNN3 (0.46) KCNN3KCNN1KCNN2PDE10ACDK2
SCHEMBL7447428 0.83 CYP1A2 (0.44) KCNN3KCNN1KCNN2CDK2CCNE1
SCHEMBL7441328 0.79 KCNN3 (0.62) KCNN3KCNN1KCNN2PDE10ACDK2
SCHEMBL7441150 0.77 CDK2 (0.48) CDK2CCNE1MEN1USP2ALDH1A1
SCHEMBL13117302 0.76 KCNN3 (0.80) KCNN3KCNN1KCNN2PDE10ACDK2
SCHEMBL7445599 0.75 DPP4 (0.42) KCNN3KCNN1KCNN2PDE10AALDH1A1
SCHEMBL7436471 0.75 MYC (0.40) MEN1USP2ALDH1A1CYP1A2CYP3A4
SCHEMBL30083383 0.74 CDK2 (0.67) KCNN3KCNN1KCNN2CDK2CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed