SCHEMBL7435705

SCHEMBL7435705

CCCCc1cc(NCc2ccc(-c3ccccc3C#N)cc2)n2nccc2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN3 Q9UGI6 5/20 0.46
KCNN1 Q92952 1/20 0.46
KCNN2 Q9H2S1 1/20 0.46
CCNT1 O60563 1/20 0.44
CDK7 P50613 1/20 0.44
CDK9 P50750 1/20 0.44
CCNH P51946 1/20 0.44
PRKAB2 O43741 1/20 0.43
PRKAG1 P54619 1/20 0.43
PRKAA2 P54646 1/20 0.43
PRKAA1 Q13131 1/20 0.43
PRKAG3 Q9UGI9 1/20 0.43
PRKAG2 Q9UGJ0 1/20 0.43
PRKAB1 Q9Y478 1/20 0.43
CDK2 P24941 6/20 0.43
ACHE P22303 1/20 0.43
CCNE1 P24864 4/20 0.42
PPARG P37231 2/20 0.42
AGTR1 P30556 1/20 0.40
PDE10A Q9Y233 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7437667 0.91 PRKAB2 (0.51) KCNN3KCNN1KCNN2PRKAB2PRKAG1
SCHEMBL7441417 0.84 MEN1 (0.49) KCNN3KCNN1KCNN2CDK2CCNE1
SCHEMBL7445604 0.84 KCNN3 (0.66) KCNN3KCNN1KCNN2CDK2CCNE1
SCHEMBL7442662 0.80 KCNN3 (0.45) KCNN3KCNN1KCNN2CCNT1CDK7
SCHEMBL7435695 0.80 DPP4 (0.39) CCNT1CDK7CDK9CCNHCDK2
SCHEMBL7449214 0.79 CDK2 (0.46) CDK2CCNE1PPARGAGTR1
SCHEMBL7447428 0.78 CYP1A2 (0.44) KCNN3KCNN1KCNN2CDK9PRKAG1
SCHEMBL7445484 0.78 PRKAB2 (0.42) KCNN3KCNN1KCNN2CDK7CDK9
SCHEMBL7447205 0.76 CDK2 (0.46) CDK2ACHECCNE1PPARG
SCHEMBL7447111 0.76 GAA (0.51) CDK2PPARGMYCWDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed