SCHEMBL7445637

SCHEMBL7445637

CCOC(=O)CN(C(=O)Oc1ccc2[nH]c(CNc3ccc(C#N)cc3)nc2c1C)c1ccccn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39
NQO2 P16083 1/20 0.36
TGFBR1 P36897 5/20 0.33
POLB P06746 2/20 0.33
CHEK1 O14757 1/20 0.33
IDH1 O75874 1/20 0.32
PIP4K2A P48426 1/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
NR1I2 O75469 1/20 0.32
F2 P00734 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
SLC6A2 P23975 1/20 0.32
AGTR1 P30556 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7444335 0.89 MAPT (0.41) ALDH1A1NPC1LMNAMAPTMAPK1
Hydrochloric Acid SCHEMBL7444749 0.88 NQO2 (0.47) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL7448239 0.85 POLB (0.33) ALDH1A1MAPTNQO2POLBMEN1
SCHEMBL9901721 0.84 NQO2 (0.46) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL7444535 0.82 ALDH1A1 (0.40) ALDH1A1NPC1LMNAMAPTMAPK1
Acetic Acid SCHEMBL17065511 0.82 NQO2 (0.45) ALDH1A1NPC1LMNAMAPTMAPK1
Hydrochloric Acid SCHEMBL7444759 0.81 KLK1 (0.44) ALDH1A1NPC1LMNAMAPTMAPK1
Hydrochloric Acid SCHEMBL7454281 0.81 KLK1 (0.44) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL7452770 0.81 HCRTR1 (0.34) ALDH1A1MAPTMAPK1NQO2CHEK1
Hydrochloric Acid SCHEMBL7447095 0.81 NQO2 (0.54) ALDH1A1NPC1LMNAMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966454-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS Boehringer Ingelheim Pharma KG (DE) 1999-12-29 EP disclosed
WO-1998037075-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-08-27 WO disclosed