SCHEMBL7445980

SCHEMBL7445980

CCOC(=O)Cc1c(OS(=O)(=O)C(F)(F)F)cc(C)[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.42
MAPK1 P28482 2/20 0.42
USP2 O75604 1/20 0.42
TSHR P16473 1/20 0.42
KDM4E B2RXH2 7/20 0.40
LMNA P02545 3/20 0.40
ALDH1A1 P00352 3/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
L3MBTL1 Q9Y468 3/20 0.37
GLA P06280 2/20 0.37
ATM Q13315 2/20 0.37
CASP1 P29466 2/20 0.37
CASP7 P55210 2/20 0.37
MAPT P10636 1/20 0.37
THRB P10828 1/20 0.37
HTT P42858 1/20 0.37
GAA P10253 2/20 0.36
EZH2 Q15910 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7451513 0.74 KDM4E (0.59) HSD17B10MAPK1USP2TSHRKDM4E
SCHEMBL7440362 0.72 MAPK1 (0.38) HSD17B10MAPK1USP2TSHRKDM4E
SCHEMBL14252745 0.72 SMN1; SMN2 (0.40) HSD17B10TSHRKDM4ELMNAALDH1A1
SCHEMBL2905044 0.71 SMN1; SMN2 (0.38) HSD17B10MAPK1TSHRKDM4ELMNA
SCHEMBL28138436 0.71 SMN1; SMN2 (0.40) HSD17B10MAPK1TSHRKDM4ELMNA
SCHEMBL28166901 0.70 ABL1 (0.42) HSD17B10TSHRKDM4ELMNAALDH1A1
SCHEMBL3718701 0.70 CA5A (0.54) TSHRALDH1A1KMT2ATDP1SMN1; SMN2
SCHEMBL28167083 0.70 ABL1 (0.39) HSD17B10MAPK1TSHRKDM4ELMNA
SCHEMBL2128158 0.70 L3MBTL1 (0.35) HSD17B10MAPK1TSHRKDM4EKMT2A
SCHEMBL151254 0.70 MAPT (0.40) HSD17B10TSHRKDM4ELMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1124822-A4 THROMBIN INHIBITORS MERCK & CO INC (US) 2002-04-03 EP disclosed
EP-1124822-A1 THROMBIN INHIBITORS Merck & Co., Inc. (US) 2001-08-22 EP disclosed
WO-2000026211-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2000-05-11 WO disclosed