SCHEMBL7446643

SCHEMBL7446643

COc1ccc(CCN2CCOCC2)c(Oc2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.53
KDM1A O60341 1/20 0.51
ALDH1A1 P00352 4/20 0.50
TSHR P16473 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
KDM4E B2RXH2 1/20 0.49
MAPT P10636 1/20 0.49
SIGMAR1 Q99720 2/20 0.48
PTPN1 P18031 1/20 0.48
SLC6A4 P31645 2/20 0.47
HRH3 Q9Y5N1 1/20 0.47
HTR1A P08908 1/20 0.47
MAPK1 P28482 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
LMNA P02545 1/20 0.47
KCNH2 Q12809 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6177281 0.78 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2KDM4EMAPTL3MBTL1
SCHEMBL23926326 0.77 SIGMAR1 (0.79) TSHRSIGMAR1HRH3KCNH2
SCHEMBL30118894 0.77 SIGMAR1 (0.79) TSHRSIGMAR1HRH3KCNH2
SCHEMBL6180224 0.74 LTA4H (0.47) SMN1; SMN2KDM4ESLC6A4HTR1AKCNH2
Hydrochloric Acid SCHEMBL9644987 0.74 KCNH2 (0.80) SIGMAR1HRH3KCNH2
SCHEMBL21587706 0.73 KDM4E (0.64) ALDH1A1TSHRSMN1; SMN2KDM4EMAPT
SCHEMBL13110052 0.73 SLC6A4 (0.66) ALDH1A1KDM4ESIGMAR1SLC6A4HRH3
SCHEMBL15143993 0.73 SMN1; SMN2 (0.54) TSHRSMN1; SMN2KDM4ESIGMAR1HRH3
SCHEMBL11365451 0.71 ALDH1A1 (0.55) ALDH1A1TSHRSMN1; SMN2NPSR1KDM4E
SCHEMBL9069989 0.71 SIGMAR1 (0.77) SMN1; SMN2SIGMAR1HRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025090-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2000-11-08 EP disclosed
EP-1025090-A1 VITRONECTIN RECEPTOR ANTAGONISTS SmithKline Beecham Corporation (US) 2000-08-09 EP disclosed
WO-1999015508-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-04-01 WO disclosed