SCHEMBL7447016

SCHEMBL7447016

CCCc1cc(C(=O)c2ccsc2)ccc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALDH1A1 P00352 4/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
POLB P06746 1/20 0.43
PPARG P37231 2/20 0.42
PPARD Q03181 1/20 0.42
PPARA Q07869 1/20 0.42
TUBB4A P04350 2/20 0.42
TUBB P07437 2/20 0.42
TUBA3C P0DPH7 2/20 0.42
TUBA1B P68363 2/20 0.42
TUBA4A P68366 2/20 0.42
TUBB4B P68371 2/20 0.42
TUBB3 Q13509 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24648546 0.80 POLB (0.52) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL24648543 0.80 ALDH1A1 (0.53) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL7444751 0.79 CYP1A2 (0.53) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL7447786 0.78 ALDH1A1 (0.73) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL24648542 0.77 CYP1A2 (0.52) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL6343700 0.77 ALDH1A1 (0.65) ALDH1A1HTTL3MBTL1POLBGAA
SCHEMBL3547262 0.77 CA12 (0.61) TSHRALDH1A1LMNAHTTMEN1
SCHEMBL11575413 0.76 CYP1A2 (0.66) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL6958930 0.76 SLC22A6 (0.73) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL20058880 0.76 MAPK1 (0.60) CYP1A2CYP3A4CYP2C9TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed