SCHEMBL7447111

SCHEMBL7447111

CCc1cc(NCc2ccc(-c3ccccc3C#N)cc2)n2ncnc2n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.51
ALDH1A1 P00352 5/20 0.43
HSD17B10 Q99714 4/20 0.43
CYP1A2 P05177 4/20 0.43
CYP3A4 P08684 4/20 0.43
TSHR P16473 3/20 0.43
CYP2C9 P11712 3/20 0.43
CYP2C19 P33261 3/20 0.43
MAPK1 P28482 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CLK4 Q9HAZ1 2/20 0.43
USP2 O75604 1/20 0.43
CYP2D6 P10635 1/20 0.43
BLM P54132 1/20 0.43
KDM4E B2RXH2 4/20 0.42
HPGD P15428 4/20 0.42
ALPL P05186 1/20 0.42
ALPG P10696 1/20 0.42
CDK2 P24941 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7437667 0.84 PRKAB2 (0.51) ALDH1A1HSD17B10CYP1A2CYP3A4TSHR
SCHEMBL7439169 0.83 CYP1A2 (0.41) ALDH1A1HSD17B10CYP1A2CYP3A4TSHR
SCHEMBL7437260 0.82 CDK2 (0.49) ALDH1A1HSD17B10CYP1A2CYP3A4TSHR
SCHEMBL7441150 0.81 CDK2 (0.48) ALDH1A1HSD17B10CYP1A2CYP3A4TSHR
SCHEMBL7449214 0.80 CDK2 (0.46) GAAALDH1A1HSD17B10CYP1A2CYP3A4
SCHEMBL7446034 0.80 GAA (0.48) GAAALDH1A1HSD17B10CYP1A2CYP3A4
SCHEMBL7447205 0.80 CDK2 (0.46) ALDH1A1HSD17B10CYP1A2CYP3A4TSHR
SCHEMBL7447121 0.78 TSHR (0.41) ALDH1A1HSD17B10CYP1A2CYP3A4TSHR
SCHEMBL7433300 0.78 CDK2 (0.44) ALDH1A1HSD17B10CYP1A2CYP3A4TSHR
SCHEMBL7435705 0.76 KCNN3 (0.46) CDK2PPARGMYCWDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed