SCHEMBL7447330

SCHEMBL7447330

CCCn1c(CCl)nc2ccc(F)cc21

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.48
AGTR2 P50052 2/20 0.48
CYP11B2 P19099 3/20 0.43
CYP11B1 P15538 2/20 0.43
RPS6KA5 O75582 1/20 0.42
RAB9A P51151 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
PKM P14618 1/20 0.41
BRD4 O60885 1/20 0.40
TP53 P04637 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPT P10636 1/20 0.38
KDM4E B2RXH2 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5109530 0.88 AGTR1 (0.48) AGTR1AGTR2RPS6KA5RAB9AMEN1
Bromide SCHEMBL5929370 0.87 AGTR1 (0.47) AGTR1AGTR2RPS6KA5RAB9AMEN1
SCHEMBL13872476 0.80 CYP11B2 (0.49) AGTR1AGTR2CYP11B2CYP11B1RPS6KA5
SCHEMBL7019632 0.79 CYP11B2 (0.47) CYP11B2CYP11B1RAB9AMEN1KMT2A
SCHEMBL3059715 0.78 MEN1 (0.64) RAB9AMEN1KMT2APKMTP53
Hydrochloric Acid SCHEMBL7015191 0.78 CYP11B2 (0.46) CYP11B2CYP11B1RAB9AMEN1KMT2A
SCHEMBL28952848 0.75 AGTR1 (0.38) AGTR1AGTR2CYP11B2CYP11B1RPS6KA5
SCHEMBL5096807 0.73 AGTR1 (0.46) AGTR1AGTR2RPS6KA5RAB9AMEN1
SCHEMBL7745377 0.73 TSHR (0.50) AGTR1AGTR2
SCHEMBL13274084 0.73 PPARG (0.47) RAB9AKMT2ATP53ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165557-A1 ARYL AND HETEROARYL FUSED AMINOALKYL-IMIDAZOLE DERIVATIVES: SELECTIVE MODULATORS OF GABAa RECEPTORS NEUROGEN CORPORATION (US) 2002-01-02 EP disclosed
WO-2000059905-A1 ARYL AND HETEROARYL FUSED AMINOALKYL-IMIDAZOLE DERIVATIVES: SELECTIVE MODULATORS OF GABAa RECEPTORS NEUROGEN CORPORATION (US) 2000-10-12 WO disclosed