SCHEMBL7019632

SCHEMBL7019632

CCCn1c(CCl)nc2ccc(C#N)cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 4/20 0.47
ACSS2 Q9NR19 1/20 0.46
CYP11B1 P15538 3/20 0.45
BRD4 O60885 1/20 0.43
DAPK3 O43293 1/20 0.38
MAP4K4 O95819 1/20 0.38
PRKACA P17612 1/20 0.38
LTK P29376 1/20 0.38
MAPK8 P45983 1/20 0.38
CSNK1A1 P48729 1/20 0.38
CDK8 P49336 1/20 0.38
CLK2 P49760 1/20 0.38
CDK9 P50750 1/20 0.38
LIMK1 P53667 1/20 0.38
CDK5 Q00535 1/20 0.38
MAP2K1 Q02750 1/20 0.38
LRRK2 Q5S007 1/20 0.38
AURKB Q96GD4 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
ALK Q9UM73 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7015191 0.99 CYP11B2 (0.46) CYP11B2ACSS2CYP11B1BRD4DAPK3
SCHEMBL3061472 0.89 ALOX5AP (0.43) MEN1KMT2AALOX5AP
Hydrochloric Acid SCHEMBL3063212 0.88 ALOX5AP (0.42) MEN1KMT2AALOX5AP
SCHEMBL6218225 0.86 TSHR (0.47) CYP11B2ACSS2CYP11B1BRD4DAPK3
SCHEMBL1161796 0.83 PPARG (0.46) CYP11B2ACSS2CYP11B1BRD4DAPK3
SCHEMBL1638406 0.82 ACSS2 (0.43) CYP11B2ACSS2CYP11B1BRD4LMNA
SCHEMBL1638450 0.80 MAPT (0.47) CYP11B2ACSS2CYP11B1BRD4LMNA
SCHEMBL1638650 0.80 ACSS2 (0.42) CYP11B2ACSS2CYP11B1BRD4LMNA
SCHEMBL7447330 0.79 AGTR1 (0.48) CYP11B2CYP11B1BRD4MEN1KMT2A
SCHEMBL1636416 0.78 ACSS2 (0.40) CYP11B2ACSS2CYP11B1BRD4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368342-A2 BENZIMIDAZOLE AND PYRIDYLIMIDAZOLE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS NEUROGEN CORPORATION (US) 2003-12-10 EP disclosed
WO-2002050062-A2 BENZIMIDAZOLE AND PYRIDYLIMIDAZOLE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS NEUROGEN CORPORATION (US) 2002-06-27 WO disclosed