SCHEMBL7447432

SCHEMBL7447432

O=c1cc(-c2ccncc2)[nH]c(N2CCCCC2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.47
PKN1 Q16512 2/20 0.46
PKN2 Q16513 2/20 0.46
CDC7 O00311 8/20 0.43
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
ADORA1 P30542 1/20 0.41
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
CDK9 P50750 3/20 0.40
HPGD P15428 2/20 0.40
DYRK3 O43781 2/20 0.40
ROCK2 O75116 2/20 0.40
CDK1 P06493 2/20 0.40
PRKACA P17612 2/20 0.40
CDK2 P24941 2/20 0.40
MAPK1 P28482 2/20 0.40
CSNK1A1 P48729 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5386406 0.99 HSD17B10 (0.45) HSD17B10PKN1PKN2CDC7MEN1
SCHEMBL5381026 0.86 AR (0.44) HSD17B10CDC7MEN1KMT2ACDK2
SCHEMBL7978699 0.81 MAPT (0.52) HSD17B10CDC7MEN1CYP1A2CYP2C19
SCHEMBL7989788 0.79 ALDH1A1 (0.58) HSD17B10MEN1CYP2C19KMT2AHPGD
SCHEMBL7990353 0.78 KDM4E (0.52) HSD17B10CYP1A2HPGDMAPK1KDM4E
SCHEMBL7990765 0.78 CDC7 (0.39) PKN1PKN2CDC7CDK9DYRK3
SCHEMBL7978276 0.77 HRH4 (0.49)
SCHEMBL5380085 0.77 HSD17B10 (0.77) HSD17B10CDC7MEN1CYP1A2CYP2C19
SCHEMBL7989669 0.76 KCNH2 (0.35) CDC7
SCHEMBL7978711 0.76 POLB (0.46) HSD17B10GSK3BKDM4EALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115721-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP disclosed
WO-2000018758-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2000-04-06 WO disclosed