SCHEMBL7447626

SCHEMBL7447626

COc1cc(C(=O)C(=O)O)ccc1OCCCN1CCC(=C(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.47
CHRM2 P08172 1/20 0.47
HTR1A P08908 1/20 0.47
ADRA2A P08913 1/20 0.47
CHRM1 P11229 1/20 0.47
DRD2 P14416 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
DRD1 P21728 1/20 0.47
DRD4 P21917 1/20 0.47
ACHE P22303 1/20 0.47
SLC6A2 P23975 1/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
SLC6A4 P31645 1/20 0.47
CCKBR P32239 1/20 0.47
ADRA1A P35348 1/20 0.47
HRH1 P35367 1/20 0.47
OPRM1 P35372 1/20 0.47
DRD3 P35462 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430589 0.95 ABCB11 (0.44) ABCB11CHRM2HTR1AADRA2ACHRM1
SCHEMBL7441629 0.92 KDM4E (0.49) ACHEOPRM1KDM4ETDP1ALDH1A1
Oxalic Acid SCHEMBL10459130 0.91 ABCB11 (0.55) ABCB11CHRM2HTR1AADRA2ACHRM1
SCHEMBL10562079 0.90 ABCB11 (0.57) ABCB11CHRM2HTR1AADRA2ACHRM1
Oxalic Acid SCHEMBL10461881 0.89 KDM4E (0.56) ABCB11CHRM2HTR1AADRA2ACHRM1
SCHEMBL10559960 0.89 OPRM1 (0.54) ABCB11CHRM2HTR1AADRA2ACHRM1
Oxalic Acid SCHEMBL10460875 0.88 KDM4E (0.57) DRD2DRD4HTR2AHTR2COPRM1
Oxalic Acid SCHEMBL10460394 0.86 DRD3 (0.52) DRD2DRD4HRH1DRD3KDM4E
SCHEMBL7443832 0.85 ABCB11 (0.43) ABCB11CHRM2HTR1AADRA2ACHRM1
SCHEMBL10559200 0.84 ALDH1A1 (0.48) HTR1ADRD2DRD3KDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5070087-A Aryl(alkyland alkylene)-N-((phenoxy and phenylthio)alkyl) aminoheterocyclics as cardiovascular, anthihistaminic, antisecretory and antiallergy agents A. H. ROBINS COMPANY, INCORPORATED (US) 1991-12-03 US disclosed