SCHEMBL7447749

SCHEMBL7447749

CC(C)(C)c1ccc(CN(Cc2ccc(C(C)(C)C)cc2)[C@@H](Cc2ccc(OCc3ccccc3)cc2)C(=O)NCCN2CCCCC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
EPOR P19235 9/20 0.50
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
EGFR P00533 2/20 0.46
KDM4E B2RXH2 2/20 0.46
NPY1R P25929 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
HTT P42858 1/20 0.46
TACR2 P21452 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447767 1.00 ALDH1A1 (0.52) ALDH1A1EPORNPC1RAB9ASMN1; SMN2
SCHEMBL7455621 0.84 ALDH1A1 (0.52) ALDH1A1NPC1RAB9ASMN1; SMN2EGFR
SCHEMBL7450350 0.84 ALDH1A1 (0.52) ALDH1A1NPC1RAB9ASMN1; SMN2EGFR
SCHEMBL7454928 0.83 HRH3 (0.46) ALDH1A1NPC1RAB9ASMN1; SMN2EGFR
SCHEMBL8193049 0.82 CTSS (0.48) ALDH1A1TACR2
SCHEMBL7365328 0.79 NPC1 (0.56) ALDH1A1NPC1RAB9ASMN1; SMN2EGFR
SCHEMBL7341842 0.79 NPC1 (0.56) ALDH1A1NPC1RAB9ASMN1; SMN2EGFR
SCHEMBL7371156 0.78 HTT (0.57) ALDH1A1NPC1RAB9ASMN1; SMN2EGFR
SCHEMBL7446328 0.78 AKT1 (0.60) TACR2
SCHEMBL7344798 0.76 TACR2 (0.53) NPC1RAB9ASMN1; SMN2TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6180677-B1 ANTIEPILEPSY AGENT WARNER-LAMBERT COMPANY 2001-01-30 US claimed
WO-2000006535-A1 TYROSINE-DERIVED COMPOUNDS AS CALCIUM CHANNEL ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2000-02-10 WO claimed
US-6323243-B1 AROMATIC ETHER WITH AMINE OR AMIDE GROUPS WARNER-LAMBERT COMPANY 2001-11-27 US disclosed
US-6180677-B1 ANTIEPILEPSY AGENT WARNER-LAMBERT COMPANY 2001-01-30 US disclosed
WO-2000006535-A1 TYROSINE-DERIVED COMPOUNDS AS CALCIUM CHANNEL ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2000-02-10 WO disclosed