SCHEMBL7447927

SCHEMBL7447927

CC(=O)Oc1ccc2c(c1OC(C)=O)CC(c1ccccc1)C=C2CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.38
ATM Q13315 1/20 0.38
BACE1 P56817 12/20 0.38
BUB1 O43683 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447921 1.00 KMT2A (0.38) KMT2AATMBACE1BUB1
Hydrochloric Acid SCHEMBL7440754 0.99 KMT2A (0.37) KMT2AATMBACE1BUB1
Hydrochloric Acid SCHEMBL7440751 0.99 KMT2A (0.37) KMT2AATMBACE1BUB1
Hydrochloric Acid SCHEMBL7447474 0.89 DRD2 (0.35) KMT2A
SCHEMBL7449625 0.89 MASP2 (0.34)
Hydrochloric Acid SCHEMBL8829325 0.88 MASP2 (0.33)
Hydrochloric Acid SCHEMBL8829320 0.88 MASP2 (0.33)
SCHEMBL7444849 0.84 CARM1 (0.36) BACE1
SCHEMBL7444847 0.84 CARM1 (0.36) BACE1
SCHEMBL7443351 0.82 ADORA3 (0.36) KMT2AATMBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5621133-A PREPARING A 1-(3,4-DIALKOXYPHENYL),3-HYDROXYALKANE(C6-C12) BY EPOXIDIZING A HALO DERIVATIVE WITH A BASE FOLLOWED BY DECYCLICIZING WITH AN ORGANOMETALLIC COMPOUND IN A SOLVENT; NAPHTHYLENES, ISOCHROMENES AND ISOTHIOCHROMENES DENINNO MICHAEL P (US) 1997-04-15 US disclosed
US-5591884-A PROTECTED HYDROXYALKYLCATECHOL INTERMEDIATES ABBOTT LABORATORIES (US) 1997-01-07 US disclosed
WO-1996038435-A1 DOPAMINE AGONISTS ABBOTT LABORATORIES (US) 1996-12-05 WO disclosed
EP-0474767-B1 DOPAMINE AGONISTS ABBOTT LAB (US) 1996-02-21 EP disclosed