SCHEMBL7448203

SCHEMBL7448203

NC(=O)CCCc1cc(F)ccc1F

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 7/20 0.57
SLC6A4 P31645 1/20 0.57
MAPK8 P45983 2/20 0.43
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
RIPK1 Q13546 1/20 0.41
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40
GABRA2 P47869 1/20 0.40
GABRB2 P47870 1/20 0.40
GABRA4 P48169 1/20 0.40
GABRE P78334 1/20 0.40
GABRA6 Q16445 1/20 0.40
GABRG1 Q8N1C3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9160653 0.87 MPO (0.59) MPOSLC6A4MAPK8CES2CES1
SCHEMBL8240809 0.86 PSEN1 (0.47) MPOSLC6A4CES2CES1DPP4
SCHEMBL9955740 0.83 DGAT1 (0.46) MPOSLC6A4MTNR1ATLR8
SCHEMBL8239860 0.81 F13A1 (0.53) MPOCES2CES1RIPK1DPP4
SCHEMBL9160970 0.80 MPO (0.56) MPOSLC6A4MAPK8CES2CES1
SCHEMBL28038980 0.79 CES2 (0.45) MPOSLC6A4MAPK8CES2CES1
SCHEMBL1115079 0.79 MAPK8 (0.52) MPOSLC6A4MAPK8CES2CES1
SCHEMBL29009856 0.79 F13A1 (0.56) MPOMAPTPSEN1PSEN2APH1B
SCHEMBL1478187 0.78 FFAR1 (0.51) CES2CES1
SCHEMBL5261311 0.78 MPO (0.56) MPOSLC6A4MTNR1ATLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002541151-A 2002-12-03 JP claimed
EP-1165557-A1 ARYL AND HETEROARYL FUSED AMINOALKYL-IMIDAZOLE DERIVATIVES: SELECTIVE MODULATORS OF GABAa RECEPTORS NEUROGEN CORPORATION (US) 2002-01-02 EP claimed
WO-2000059905-A1 ARYL AND HETEROARYL FUSED AMINOALKYL-IMIDAZOLE DERIVATIVES: SELECTIVE MODULATORS OF GABAa RECEPTORS NEUROGEN CORPORATION (US) 2000-10-12 WO claimed