SCHEMBL7448204

SCHEMBL7448204

CCCN(CCC)C1Cc2cc3c(cc2C1)C(=O)N(Cc1ccc(C#N)cc1)C3=O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FYN P06241 1/20 0.42
HTR1A P08908 1/20 0.42
DRD3 P35462 1/20 0.41
ADRA1D P25100 2/20 0.41
ADRA1A P35348 2/20 0.41
ADRA1B P35368 2/20 0.41
ALDH1A1 P00352 3/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
GAA P10253 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
ALOX12 P18054 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7456278 0.86 DRD3 (0.50) FYNHTR1ADRD3ALDH1A1CYP2D6
SCHEMBL7457771 0.85 FNTA (0.40) FYNHTR1ADRD3ALDH1A1CYP2D6
SCHEMBL7451624 0.85 FYN (0.45) FYNHTR1ADRD3ALDH1A1CYP2D6
SCHEMBL8103965 0.85 ALDH1A1 (0.55) FYNHTR1ADRD3ALDH1A1CYP2D6
SCHEMBL7453175 0.84 FYN (0.44) FYNHTR1ADRD3ALDH1A1CYP2D6
SCHEMBL7451238 0.83 DRD2 (0.51) DRD3ALDH1A1CYP2D6CYP2C9ALOX15
SCHEMBL7443295 0.83 FYN (0.45) FYNHTR1ADRD3ALDH1A1CYP2D6
SCHEMBL7456265 0.81 DRD3 (0.54) FYNHTR1ADRD3ALDH1A1CYP2D6
SCHEMBL7456004 0.81 CA1 (0.56) FYNHTR1ADRD3
SCHEMBL8103977 0.80 FYN (0.55) FYNHTR1ADRD3ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6084130-A FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS PHARMACIA & UPJOHN COMPANY (US) 2000-07-04 US disclosed
EP-0923542-A1 ARYL SUBSTITUTED CYCLIC AMINES AS SELECTIVE DOPAMINE D3 LIGANDS PHARMACIA & UPJOHN COMPANY (US) 1999-06-23 EP disclosed
WO-1997045403-A1 ARYL SUBSTITUTED CYCLIC AMINES AS SELECTIVE DOPAMINE D3 LIGANDS PHARMACIA & UPJOHN COMPANY (US) 1997-12-04 WO disclosed