SCHEMBL7448247

SCHEMBL7448247

CC1(c2cccc(C#N)c2)OC1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.45
BACE1 P56817 1/20 0.39
NOTUM Q6P988 2/20 0.39
ENPP2 Q13822 1/20 0.38
VNN1 O95497 2/20 0.38
ALDH1A1 P00352 2/20 0.38
CNR2 P34972 1/20 0.38
GRIN2B Q13224 1/20 0.37
GSK3B P49841 2/20 0.37
XDH P47989 1/20 0.37
SLC22A12 Q96S37 1/20 0.37
NSD2 O96028 1/20 0.36
GRM5 P41594 1/20 0.36
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18316474 0.78 CRHBP (0.44) HSD11B1ALDH1A1MEN1MAPTKMT2A
SCHEMBL2234611 0.78 CRHBP (0.44) HSD11B1ALDH1A1MEN1MAPTKMT2A
SCHEMBL27475218 0.70 HSD11B1 (0.44) HSD11B1BACE1NOTUMALDH1A1CNR2
SCHEMBL3107917 0.69 HCAR2 (0.72)
Bicarbonate SCHEMBL11598627 0.68 GSK3B (0.55) NOTUMENPP2ALDH1A1GSK3BXDH
SCHEMBL10083343 0.68 HSD11B1 (0.50) HSD11B1VNN1ALDH1A1CNR2GRIN2B
SCHEMBL11833782 0.68 CRHBP (0.41) MEN1KMT2A
SCHEMBL16954195 0.68 HSD11B1 (0.42) HSD11B1BACE1VNN1ALDH1A1CNR2
Bicarbonate SCHEMBL28730324 0.66 GSK3B (0.53) NOTUMENPP2ALDH1A1GSK3BXDH
SCHEMBL29793755 0.66 ICMT (0.43) HSD11B1BACE1ENPP2NSD2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189879-A1 INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2002-03-27 EP disclosed
WO-2000071512-A1 INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2000-11-30 WO disclosed