SCHEMBL7449096

SCHEMBL7449096

O=C(CN1Cc2ccccc2C[C@H](N2C(=O)c3ccccc3C2=O)C1=O)OC(c1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.40
ACE P12821 3/20 0.38
MME P08473 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
RECQL P46063 1/20 0.37
ALOX15 P16050 3/20 0.37
KDM4E B2RXH2 2/20 0.37
TSHR P16473 2/20 0.37
SIRT1 Q96EB6 1/20 0.37
GAA P10253 1/20 0.36
ALDH1A1 P00352 2/20 0.36
XIAP P98170 1/20 0.36
HKDC1 Q2TB90 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KMT2A Q03164 4/20 0.36
MEN1 O00255 3/20 0.36
TAAR1 Q96RJ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7449087 1.00 HRH4 (0.40) HRH4ACEMMECYP3A4CYP2C19
SCHEMBL7357061 0.83 ACE (0.49) ACEMMEALOX15KDM4ETSHR
SCHEMBL3865826 0.83 ACE (0.49) ACEMMEALOX15KDM4ETSHR
SCHEMBL7443272 0.82 HRH4 (0.42) HRH4ACEMMEGAA
SCHEMBL7443268 0.82 HRH4 (0.42) HRH4ACEMMEGAA
SCHEMBL7441321 0.79 THRB (0.40) CYP3A4CYP2C19ALOX15KDM4ETSHR
SCHEMBL7501387 0.71 ALOX15 (0.43) MMECYP3A4CYP2C19ALOX15KDM4E
SCHEMBL8212856 0.71 ALOX15 (0.43) MMECYP3A4CYP2C19ALOX15KDM4E
SCHEMBL7450646 0.70 HRH4 (0.57) HRH4ACEMME
SCHEMBL7450649 0.70 HRH4 (0.57) HRH4ACEMME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994026719-A1 MERCAPTO-AMIDE DERIVATIVES USEFUL AS NEUTRAL ENDOPEPTIDASE AND ACE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-11-24 WO disclosed