SCHEMBL7449396

SCHEMBL7449396

CCOC(=O)CCC(=O)N(C1CCCC1)C1(c2ccc3[nH]c(CCNc4ccc(C#N)cc4)nc3c2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.37
KDM4E B2RXH2 3/20 0.35
TNKS O95271 2/20 0.33
PARP1 P09874 2/20 0.33
PARP2 Q9UGN5 2/20 0.33
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33
PLG P00747 1/20 0.33
PRSS1 P07477 1/20 0.33
PRSS2 P07478 1/20 0.33
PRSS3 P35030 1/20 0.33
PIN1 Q13526 1/20 0.33
ALDH1A1 P00352 3/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7413025 0.80 F2 (0.43) KDM4EF2F10PLGPRSS1
SCHEMBL7449392 0.79 NPC1 (0.34) MAPTTNKSPARP1PARP2ALDH1A1
SCHEMBL7450500 0.73 MLLT1 (0.39) MAPTF2F10ALDH1A1NPC1
SCHEMBL7413022 0.73 F2 (0.43) F2F10PLGPRSS1PRSS2
SCHEMBL7445649 0.71 MLLT1 (0.37) MAPTF2F10PIN1ALDH1A1
SCHEMBL7446447 0.70 F2 (0.40) MAPTTNKSPARP1PARP2F2
SCHEMBL12618999 0.70 MAPT (0.65) MAPTKDM4EPIN1ALDH1A1CYP1A2
SCHEMBL7414205 0.70 F2 (0.31) F2F10PLGPRSS1PRSS2
SCHEMBL7414208 0.70 CYP11B2 (0.33) KDM4EF2F10PLGPRSS1
SCHEMBL27553886 0.69 FASN (0.34) F2F10PLGPRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095025-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-05-02 EP disclosed
WO-2000001704-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-01-13 WO disclosed