SCHEMBL7449528

SCHEMBL7449528

CC(C)CC(NC(=O)c1ccc(N)nc1)C(=O)N(C)C#N

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSB P07858 12/20 0.53
CTSL P07711 12/20 0.48
CTSS P25774 8/20 0.48
CTSK P43235 8/20 0.48
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CA2 P00918 2/20 0.40
CA1 P00915 1/20 0.40
EPHX2 P34913 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5924957 0.88 CTSB (0.54) CTSBCTSLCTSSCTSK
SCHEMBL6183805 0.85 CTSB (0.61) CTSBCTSLCTSSCTSKCA2
SCHEMBL6182791 0.85 CTSB (0.61) CTSBCTSLCTSSCTSKCA2
SCHEMBL6183809 0.85 CTSB (0.61) CTSBCTSLCTSSCTSKCA2
SCHEMBL6182874 0.82 CTSB (0.61) CTSBCTSLCTSSCTSKCA2
SCHEMBL7132702 0.82 CTSB (0.48) CTSBCTSLCTSSCTSK
SCHEMBL5924641 0.81 CTSB (0.49) CTSBCTSLCTSSCTSK
SCHEMBL6183692 0.81 CTSL (0.67) CTSBCTSLCTSSCTSK
SCHEMBL7450448 0.81 CTSB (0.58) CTSBCTSLCTSSCTSKCA2
SCHEMBL7452244 0.80 CTSB (0.61) CTSBCTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161415-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-12 EP disclosed
WO-2000055126-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed