SCHEMBL7449608

SCHEMBL7449608

CC(C)Oc1ccc(C(=O)NC(C(=O)O)c2ccc(CNC(=O)OC(C)(C)C)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.56
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
NAMPT P43490 2/20 0.48
HDAC1 Q13547 2/20 0.46
ALDH1A1 P00352 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MAPT P10636 3/20 0.43
NPSR1 Q6W5P4 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
RECQL P46063 1/20 0.43
XBP1 P17861 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
GPR55 Q9Y2T6 1/20 0.43
SDCBP O00560 1/20 0.43
SDC2 P34741 1/20 0.43
MTTP P55157 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447906 0.91 NR1H4 (0.55) NR1H4NPC1RAB9ANAMPTHDAC1
SCHEMBL7448308 0.87 HDAC1 (0.52) NAMPTHDAC1L3MBTL1SDCBPSDC2
SCHEMBL21523879 0.83 NPC1 (0.64) NR1H4NPC1RAB9ANAMPTHDAC1
SCHEMBL4687407 0.81 CTSS (0.51) NPC1RAB9AALDH1A1SMN1; SMN2MAPT
SCHEMBL4687402 0.81 CTSS (0.51) NPC1RAB9AALDH1A1SMN1; SMN2MAPT
SCHEMBL7452422 0.80 CYP1A2 (0.45) NR1H4NPC1RAB9ANAMPTHDAC1
SCHEMBL23775465 0.80 ALDH1A1 (0.58) NR1H4NPC1RAB9ANAMPTHDAC1
SCHEMBL7446916 0.79 HDAC1 (0.50) NAMPTHDAC1MAPTNPSR1L3MBTL1
SCHEMBL7457288 0.79 HDAC1 (0.53) NAMPTHDAC1L3MBTL1MEN1KMT2A
SCHEMBL7446767 0.77 HDAC1 (0.48) NAMPTHDAC1ALDH1A1MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001027096-A9 AMINOMETHYL-(HETERO)ARYL DERIVATIVES AND THEIR USE AS TRYPTASE INHIBITORS PROTHERICS MOLECULAR DESIGN LT (GB) 2001-07-12 WO disclosed