SCHEMBL7450360

SCHEMBL7450360

O=C(O)C(=C1CSc2cc(F)c(Cl)cc2N1)[N+](=O)[O-]

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7450349 1.00 HTT (0.31) HTTKDM4EALDH1A1MAPTTDP1
SCHEMBL7451388 0.81 HTT (0.39) HTTKDM4EALDH1A1MAPTTDP1
SCHEMBL7451376 0.81 HTT (0.39) HTTKDM4EALDH1A1MAPTTDP1
SCHEMBL7454353 0.80 NOX1 (0.35) HTTKDM4EALDH1A1MAPTTDP1
SCHEMBL7453222 0.80 NPC1 (0.35) HTTKDM4EALDH1A1MAPTTDP1
SCHEMBL7451326 0.76 ALDH1A1 (0.43) HTTKDM4EALDH1A1MAPTTDP1
SCHEMBL7451322 0.76 ALDH1A1 (0.43) HTTKDM4EALDH1A1MAPTTDP1
SCHEMBL7451837 0.70 MAOA (0.47) HTTALDH1A1
SCHEMBL30954132 0.70 MAOA (0.47) HTTALDH1A1
SCHEMBL7450795 0.67 ALDH1A1 (0.47) ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151361-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-12-08 WO disclosed