SCHEMBL7450800

SCHEMBL7450800

[NH]C(=O)C([C]=O)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SRC P12931 2/20 0.43
CYP2D6 P10635 1/20 0.43
HDAC1 Q13547 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
LMNA P02545 4/20 0.41
MAPK1 P28482 1/20 0.41
CTSD P07339 1/20 0.41
CES2 O00748 2/20 0.40
CES1 P23141 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28245619 0.82 SRC (0.52) TDP1L3MBTL1SRCCYP2D6HDAC1
SCHEMBL7773819 0.82 SRC (0.52) TDP1L3MBTL1SRCCYP2D6HDAC1
SCHEMBL5609578 0.78 EPHX1 (0.46) TDP1L3MBTL1SRCCYP2D6HDAC1
SCHEMBL3237992 0.78 TDP1 (0.43) TDP1L3MBTL1SRCCYP2D6HDAC1
SCHEMBL9526813 0.77 L3MBTL1 (0.63) TDP1L3MBTL1SRCCYP2D6HDAC1
SCHEMBL3921899 0.77 CTSD (0.39) TDP1L3MBTL1SRCCYP2D6HDAC1
SCHEMBL5599310 0.77 L3MBTL1 (0.63) TDP1L3MBTL1SRCCYP2D6HDAC1
SCHEMBL1383207 0.77 TDP1 (0.56) TDP1L3MBTL1SRCCYP2D6HDAC1
SCHEMBL11341745 0.75 HDAC3 (0.44) TDP1L3MBTL1SRCCYP2D6HDAC1
SCHEMBL6596397 0.74 CYP1A2 (0.50) TDP1L3MBTL1SRCCYP2D6HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001087842-A1 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL PYRIDONES USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE PHARMACIA CORPORATION (US) 2001-11-22 WO claimed
US-4992544-A Intermediates for b-lactam antibiotics and b-lactamase inhibitor UNIVERSITY OF NOTRE DAME DU LAC (US) 1991-02-12 US disclosed